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TargetAdenosine receptor A3
LigandBDBM85776
Substrate/Competitorn/a
Ki 1704.78±n/a nM
CommentsPDSP_2057
Citation Durand, IHGreen, RD Cloning of a chick A3 adenosine receptor: characterization of ligand binding and receptor-effector coupling of chick A1 and A3 adenosine receptors. Naunyn Schmiedebergs Arch Pharmacol363:81-6 (2001) [PubMed]  Article
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Adenosine receptor A3
Name:Adenosine receptor A3
Synonyms:ADENOSINE A3 | ADORA3
Type:Enzyme Catalytic Domain
Mol. Mass.:37723.59
Organism:Chick
Description:A0A8V1ACC1
Residue:338
Sequence:
MCPQGSPCPASSSPINVTFNTSQVMGSIDVIYISAECLVALLAALGNIPVVWAVKLNAAF
HNTTMYFIASLALADIAVGVFVVPLAVLVSLQVSIPFHFCLFLCCLMVVFTQASILSLLA
IAIDRYLRVKLPIRYKIISTERRIWGALGLCWSLSLLVGLTPMFGWNKQRSAPYHTCGFT
SVIRMDYMVYFSFFAWTLIPLSIMCALYVAVFYIIRTKLSQGATGARGAGTFYGKEFRKA
KSLALILFLFAVSWLPLCIMNCVLYFHPEYKIPKPWIFLGILLSHANSAMNPVVYACKIK
KFKTTYLLILRTYILCRKKPQAMPSSYRLNTPAVVDTE
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  Blast E-value cutoff:
BDBM85776
n/a
NameBDBM85776
Synonyms:CAS_393594 | CHEMBL89852 | MRS1191 | NSC_393594
TypeSmall organic molecule
Emp. Form.C31H27NO4
Mol. Mass.477.5504
SMILESCCOC(=O)C1C(C#Cc2ccccc2)C(C(=O)OCc2ccccc2)=C(N=C1C)c1ccccc1 |c:27,29|
Structure
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