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Reaction Details
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TargetNorepinephrine transporter
LigandBDBM35226
Substrate/Competitorn/a
Ki 5.2±n/a nM
CommentsPDSP_2048
Citation Millan, MJGobert, ALejeune, FNewman-Tancredi, ARivet, JMAuclair, APeglion, JL S33005, a novel ligand at both serotonin and norepinephrine transporters: I. Receptor binding, electrophysiological, and neurochemical profile in comparison with venlafaxine, reboxetine, citalopram, and clomipramine. J Pharmacol Exp Ther298:565-80 (2001) [PubMed]
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Norepinephrine transporter
Name:Norepinephrine transporter
Synonyms:n/a
Type:Enzyme Catalytic Domain
Mol. Mass.:2082.45
Organism:RAT
Description:Norepinephrine transporter 0 RAT::Q9JIA2
Residue:19
Sequence:
MLLARMKPQVQPELGGADQ
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BDBM35226
n/a
NameBDBM35226
Synonyms:(S,S)-reboxetine | Reboxetine | Vestra
TypeSmall organic molecule
Emp. Form.C19H23NO3
Mol. Mass.313.3908
SMILESCCOc1ccccc1O[C@H]([C@@H]1CNCCO1)c1ccccc1 |r|
Structure
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