Reaction Details |
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Target | Neuropeptide Y receptor type 4 |
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Ligand | BDBM85811 |
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Substrate/Competitor | n/a |
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Ki | 5±n/a nM |
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Comments | PDSP_2037 |
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Citation | Mullins, D; Kirby, D; Hwa, J; Guzzi, M; Rivier, J; Parker, E Identification of potent and selective neuropeptide Y Y(1) receptor agonists with orexigenic activity in vivo. Mol Pharmacol60:534-40 (2001) [PubMed] |
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More Info.: | Get all data from this article |
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Neuropeptide Y receptor type 4 |
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Name: | Neuropeptide Y receptor type 4 |
Synonyms: | NPY-Y4 | NPY4-R | NPY4R | NPY4R_HUMAN | PP1 | PPYR1 | Pancreatic polypeptide receptor 1 |
Type: | Enzyme Catalytic Domain |
Mol. Mass.: | 42207.58 |
Organism: | Homo sapiens (Human) |
Description: | NPY-Y4 PPYR1 HUMAN::P50391 |
Residue: | 375 |
Sequence: | MNTSHLLALLLPKSPQGENRSKPLGTPYNFSEHCQDSVDVMVFIVTSYSIETVVGVLGNL
CLMCVTVRQKEKANVTNLLIANLAFSDFLMCLLCQPLTAVYTIMDYWIFGETLCKMSAFI
QCMSVTVSILSLVLVALERHQLIINPTGWKPSISQAYLGIVLIWVIACVLSLPFLANSIL
ENVFHKNHSKALEFLADKVVCTESWPLAHHRTIYTTFLLLFQYCLPLGFILVCYARIYRR
LQRQGRVFHKGTYSLRAGHMKQVNVVLVVMVVAFAVLWLPLHVFNSLEDWHHEAIPICHG
NLIFLVCHLLAMASTCVNPFIYGFLNTNFKKEIKALVLTCQQSAPLEESEHLPLSTVHTE
VSKGSLRLSGRSNPI
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BDBM85811 |
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n/a |
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Name | BDBM85811 |
Synonyms: | Des-AA10-17[Cys7,21, Pro34]-NPY |
Type | Small organic molecule |
Emp. Form. | C158H245N47O42S3 |
Mol. Mass. | 3571.121 |
SMILES | n/a |
Structure |
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