| Reaction Details |
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 | Report a problem with these data |
| Target | Thyrotropin-releasing hormone receptor |
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| Ligand | BDBM86217 |
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| Substrate/Competitor | n/a |
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| Ki | 3000±n/a nM |
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| Comments | PDSP_3208 |
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| Citation |  Lu, X; Bidaud, I; Ladram, A; Gershengorn, MC Pharmacological studies of thyrotropin-releasing hormone (TRH) receptors from Xenopus laevis: is xTRHR3 a TRH receptor? Endocrinology144:1842-6 (2003) [PubMed] Article |
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| More Info.: | Get all data from this article |
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| Thyrotropin-releasing hormone receptor |
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| Name: | Thyrotropin-releasing hormone receptor |
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| Synonyms: | TRHR | Thyrotropin-releasing hormone receptor 1 | thyrotropin-releasing hormone R1 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 44987.02 |
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| Organism: | Xenopus |
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| Description: | Q9DDR1 |
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| Residue: | 397 |
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| Sequence: | MDNVTFAELNATELQKREWHGLEYQVVTVFLVVVICGLGIVGNVMVVLVVLQTKHMRTPT
NCYLVSLAIADLIVLVAAGLPNITESVYGSWVYGYIGCLCITYLQYLGINASSCSITAFT
VERYLAICHPIKAQFLCTISRAKKIIVFVWAFTSLYCLMWFFLLDLNTTIYKDATVVNCG
YRVPRSYYSPIYLIDFGIFYAVPMTLATVLYGLIARILFLNPIPSDPKENSKIRKNDATH
QTKAFNSKMSSRCSNNTIASRRQVTKMLAVVVLLFAFLWMPYRTLVVVNSFLSRPYLQTW
FVLFCRICIYLNSAINPVIYNLMSQKFRAAFQKLCKCKKKRSEKPTNYGLALNYSVIKES
SNGGSPDHFSTELEDITVTDNYLSTSKMSFDDTCLPT
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| BDBM86217 |
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| n/a |
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| Name | BDBM86217 |
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| Synonyms: | Desaza1TRH |
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| Type | Small organic molecule |
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| Emp. Form. | C17H23N5O4 |
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| Mol. Mass. | 361.3956 |
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| SMILES | NC(=O)C1CCCN1C(=O)C(Cc1cnc[nH]1)NC(=O)C1CCC(=O)C1 |
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| Structure | 
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