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TargetNeuronal acetylcholine receptor subunit alpha-3
LigandBDBM50061567
Substrate/Competitorn/a
Ki 35±n/a nM
CommentsPDSP_691
Citation Xiao, YKellar, KJ The comparative pharmacology and up-regulation of rat neuronal nicotinic receptor subtype binding sites stably expressed in transfected mammalian cells. J Pharmacol Exp Ther310:98-107 (2004) [PubMed]  Article
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Neuronal acetylcholine receptor subunit alpha-3
Name:Neuronal acetylcholine receptor subunit alpha-3
Synonyms:ACHA3_RAT | Acra3 | Chrna3
Type:Enzyme
Mol. Mass.:56995.52
Organism:Rattus norvegicus (Rat)
Description:P04757
Residue:499
Sequence:
MGVVLLPPPLSMLMLVLMLLPAASASEAEHRLFQYLFEDYNEIIRPVANVSHPVIIQFEV
SMSQLVKVDEVNQIMETNLWLKQIWNDYKLKWKPSDYQGVEFMRVPAEKIWKPDIVLYNN
ADGDFQVDDKTKALLKYTGEVTWIPPAIFKSSCKIDVTYFPFDYQNCTMKFGSWSYDKAK
IDLVLIGSSMNLKDYWESGEWAIIKAPGYKHEIKYNCCEEIYQDITYSLYIRRLPLFYTI
NLIIPCLLISFLTVLVFYLPSDCGEKVTLCISVLLSLTVFLLVITETIPSTSLVIPLIGE
YLLFTMIFVTLSIVITVFVLNVHYRTPTTHTMPTWVKAVFLNLLPRVMFMTRPTSGEGDT
PKTRTFYGAELSNLNCFSRADSKSCKEGYPCQDGTCGYCHHRRVKISNFSANLTRSSSSE
SVNAVLSLSALSPEIKEAIQSVKYIAENMKAQNVAKEIQDDWKYVAMVIDRIFLWVFILV
CILGTAGLFLQPLMARDDT
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  Blast E-value cutoff:
BDBM50061567
n/a
NameBDBM50061567
Synonyms:1,1-Dimethyl-4-phenyl-piperazin-1-ium | CHEMBL134752 | CHEMBL47814 | DMPP | cid_5911
TypeSmall organic molecule
Emp. Form.C12H19N2
Mol. Mass.191.2921
SMILESC[N+]1(C)CCN(CC1)c1ccccc1
Structure
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