| Reaction Details |
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 | Report a problem with these data |
| Target | Bombesin receptor subtype-3 |
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| Ligand | BDBM86500 |
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| Substrate/Competitor | n/a |
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| Ki | 2400±n/a nM |
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| Comments | PDSP_3749 |
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| Citation |  Mantey, SA; Coy, DH; Entsuah, LK; Jensen, RT Development of bombesin analogs with conformationally restricted amino acid substitutions with enhanced selectivity for the orphan receptor human bombesin receptor subtype 3. J Pharmacol Exp Ther310:1161-70 (2004) [PubMed] Article |
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| More Info.: | Get all data from this article |
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| Bombesin receptor subtype-3 |
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| Name: | Bombesin receptor subtype-3 |
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| Synonyms: | BRS-3 | BRS3 | BRS3_HUMAN | Bombesin 3 | Bombesin like receptor 3 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 44424.45 |
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| Organism: | Homo sapiens (Human) |
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| Description: | Bombesin 3 BRS3 HUMAN::P32247 |
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| Residue: | 399 |
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| Sequence: | MAQRQPHSPNQTLISITNDTESSSSVVSNDNTNKGWSGDNSPGIEALCAIYITYAVIISV
GILGNAILIKVFFKTKSMQTVPNIFITSLAFGDLLLLLTCVPVDATHYLAEGWLFGRIGC
KVLSFIRLTSVGVSVFTLTILSADRYKAVVKPLERQPSNAILKTCVKAGCVWIVSMIFAL
PEAIFSNVYTFRDPNKNMTFESCTSYPVSKKLLQEIHSLLCFLVFYIIPLSIISVYYSLI
ARTLYKSTLNIPTEEQSHARKQIESRKRIARTVLVLVALFALCWLPNHLLYLYHSFTSQT
YVDPSAMHFIFTIFSRVLAFSNSCVNPFALYWLSKSFQKHFKAQLFCCKAERPEPPVADT
SLTTLAVMGTVPGTGSIQMSEISVTSFTGCSVKQAEDRF
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| BDBM86500 |
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| n/a |
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| Name | BDBM86500 |
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| Synonyms: | CAS_0 | NSC_0 | [D-Tyr6,Beta-Ala11,Phe13,Beta-Dap(Pr)14]Bn(6-14) |
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| Type | Small organic molecule |
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| Emp. Form. | C54H71N15O11 |
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| Mol. Mass. | 1106.2354 |
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| SMILES | CC(C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](N)Cc1ccc(O)cc1)C(=O)NCCC(=O)N[C@@H](Cc1cnc[nH]1)C(=O)N[C@@H](Cc1ccccc1)C(=O)NCC(N)C(N)=O |r| |
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| Structure | 
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