Reaction Details |
| Report a problem with these data |
Target | Promotilin |
---|
Ligand | BDBM85389 |
---|
Substrate/Competitor | n/a |
---|
Ki | 2.82±n/a nM |
---|
Comments | PDSP_6064 |
---|
Citation | Thielemans, L; Depoortere, I; Perret, J; Robberecht, P; Liu, Y; Thijs, T; Carreras, C; Burgeon, E; Peeters, TL Desensitization of the human motilin receptor by motilides. J Pharmacol Exp Ther313:1397-405 (2005) [PubMed] Article |
---|
More Info.: | Get all data from this article |
---|
|
Promotilin |
---|
Name: | Promotilin |
Synonyms: | MLN | MOTI_HUMAN | Motilin | Promotilin |
Type: | Enzyme Catalytic Domain |
Mol. Mass.: | 12919.83 |
Organism: | Homo sapiens (Human) |
Description: | Motilin 0 HUMAN::P12872 |
Residue: | 115 |
Sequence: | MVSRKAVAALLVVHVAAMLASQTEAFVPIFTYGELQRMQEKERNKGQKKSLSVWQRSGEE
GPVDPAEPIREEENEMIKLTAPLEIGMRMNSRQLEKYPATLEGLLSEMLPQHAAK
|
|
|
BDBM85389 |
---|
n/a |
---|
Name | BDBM85389 |
Synonyms: | CAS_52906-92-0 | Motilin |
Type | Small organic molecule |
Emp. Form. | C120H188N34O35S |
Mol. Mass. | 2699.049 |
SMILES | [#6]-[#6]-[#6@H](-[#6])-[#6@H](-[#7]-[#6](=O)-[#6@@H]-1-[#6]-[#6]-[#6]-[#7]-1-[#6](=O)-[#6@@H](-[#7]-[#6](=O)-[#6@@H](-[#7])-[#6]-c1ccccc1)-[#6](-[#6])-[#6])-[#6](=O)-[#7]-[#6@@H](-[#6]-c1ccccc1)-[#6](=O)-[#7]-[#6@@H](-[#6@@H](-[#6])-[#8])-[#6](=O)-[#7]-[#6@@H](-[#6]-c1ccc(-[#8])cc1)-[#6](=O)-[#7]-[#6]-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6]-[#6](-[#8])=O)-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6](-[#6])-[#6])-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6]-[#6](-[#7])=O)-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6]-[#6]\[#7]=[#6](/[#7])-[#7])-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6]-[#16]-[#6])-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6]-[#6](-[#7])=O)-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6]-[#6](-[#8])=O)-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6]-[#6]-[#6]-[#7])-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6]-[#6](-[#8])=O)-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6]-[#6]\[#7]=[#6](/[#7])-[#7])-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6](-[#7])=O)-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6]-[#6]-[#6]-[#7])-[#6](=O)-[#7]-[#6]-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6]-[#6](-[#7])=O)-[#6](-[#8])=O |r| |
Structure |
|