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TargetAdenosine receptor A2a
LigandBDBM86759
Substrate/Competitorn/a
Ki 893±n/a nM
CommentsPDSP_8525
Citation Ohshita, KIshiyama, HOyanagi, KNakata, HKobayashi, J Synthesis of hybrid molecules of caffeine and eudistomin D and its effects on adenosine receptors. Bioorg Med Chem15:3235-40 (2007) [PubMed]  Article
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Adenosine receptor A2a
Name:Adenosine receptor A2a
Synonyms:A2A adenosine receptor (hA2A) | AA2AR_HUMAN | ADENOSINE A2 | ADENOSINE A2a | ADORA2 | ADORA2A | Adenosine A2A receptor (A2AAR)
Type:G Protein-Coupled Receptor (GPCR)
Mol. Mass.:44716.46
Organism:Homo sapiens (Human)
Description:P29274
Residue:412
Sequence:
MPIMGSSVYITVELAIAVLAILGNVLVCWAVWLNSNLQNVTNYFVVSLAAADIAVGVLAI
PFAITISTGFCAACHGCLFIACFVLVLTQSSIFSLLAIAIDRYIAIRIPLRYNGLVTGTR
AKGIIAICWVLSFAIGLTPMLGWNNCGQPKEGKNHSQGCGEGQVACLFEDVVPMNYMVYF
NFFACVLVPLLLMLGVYLRIFLAARRQLKQMESQPLPGERARSTLQKEVHAAKSLAIIVG
LFALCWLPLHIINCFTFFCPDCSHAPLWLMYLAIVLSHTNSVVNPFIYAYRIREFRQTFR
KIIRSHVLRQQEPFKAAGTSARVLAAHGSDGEQVSLRLNGHPPGVWANGSAPHPERRPNG
YALGLVSGGSAQESQGNTGLPDVELLSHELKGVCPEPPGLDDPLAQDGAGVS
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  Blast E-value cutoff:
BDBM86759
n/a
NameBDBM86759
Synonyms:2,4-dimethyl-4,9-dihydro-2,4,7,9-tetraaza-fluorene-1,3-dione | CAS_44457473 | NSC_44457473
TypeSmall organic molecule
Emp. Form.C11H12N4O2
Mol. Mass.232.2386
SMILESCN1C2C(Nc3cccnc23)C(=O)N(C)C1=O
Structure
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