| Reaction Details |
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 | Report a problem with these data |
| Target | Adenosine receptor A3 |
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| Ligand | BDBM86759 |
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| Substrate/Competitor | n/a |
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| Ki | 13.90±n/a nM |
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| Comments | PDSP_8525 |
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| Citation |  Ohshita, K; Ishiyama, H; Oyanagi, K; Nakata, H; Kobayashi, J Synthesis of hybrid molecules of caffeine and eudistomin D and its effects on adenosine receptors. Bioorg Med Chem15:3235-40 (2007) [PubMed] Article |
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| More Info.: | Get all data from this article |
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| Adenosine receptor A3 |
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| Name: | Adenosine receptor A3 |
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| Synonyms: | A3 adenosine receptor (hA3) | AA3R_HUMAN | ADORA3 | Adenosine A3 receptor (A3AR) |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 36197.32 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P0DMS8 |
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| Residue: | 318 |
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| Sequence: | MPNNSTALSLANVTYITMEIFIGLCAIVGNVLVICVVKLNPSLQTTTFYFIVSLALADIA
VGVLVMPLAIVVSLGITIHFYSCLFMTCLLLIFTHASIMSLLAIAVDRYLRVKLTVRYKR
VTTHRRIWLALGLCWLVSFLVGLTPMFGWNMKLTSEYHRNVTFLSCQFVSVMRMDYMVYF
SFLTWIFIPLVVMCAIYLDIFYIIRNKLSLNLSNSKETGAFYGREFKTAKSLFLVLFLFA
LSWLPLSIINCIIYFNGEVPQLVLYMGILLSHANSMMNPIVYAYKIKKFKETYLLILKAC
VVCHPSDSLDTSIEKNSE
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| BDBM86759 |
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| n/a |
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| Name | BDBM86759 |
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| Synonyms: | 2,4-dimethyl-4,9-dihydro-2,4,7,9-tetraaza-fluorene-1,3-dione | CAS_44457473 | NSC_44457473 |
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| Type | Small organic molecule |
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| Emp. Form. | C11H12N4O2 |
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| Mol. Mass. | 232.2386 |
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| SMILES | CN1C2C(Nc3cccnc23)C(=O)N(C)C1=O |
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| Structure | 
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