| Reaction Details |
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 | Report a problem with these data |
| Target | Melanocortin receptor 4 |
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| Ligand | BDBM68044 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Luminescence-based cell-based high throughput dose response assay for biased ligands (agonists) of the melanocortin 4 receptor (MC4R) |
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| EC50 | >89205±n/a nM |
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| Citation |  PubChem, PC Luminescence-based cell-based high throughput dose response assay for biased ligands (agonists) of the melanocortin 4 receptor (MC4R) PubChem Bioassay(2012)[AID] |
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| More Info.: | Get all data from this article, Assay Method |
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| Melanocortin receptor 4 |
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| Name: | Melanocortin receptor 4 |
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| Synonyms: | MC4-R | MC4R | MC4R_HUMAN | Melanocortin MC4 | Melanocortin receptor 4 (MC-4) | Melanocortin receptor 4 (MC4-R) | Melanocortin receptor 4 (MC4R) |
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| Type: | Enzyme |
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| Mol. Mass.: | 36949.50 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P32245 |
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| Residue: | 332 |
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| Sequence: | MVNSTHRGMHTSLHLWNRSSYRLHSNASESLGKGYSDGGCYEQLFVSPEVFVTLGVISLL
ENILVIVAIAKNKNLHSPMYFFICSLAVADMLVSVSNGSETIVITLLNSTDTDAQSFTVN
IDNVIDSVICSSLLASICSLLSIAVDRYFTIFYALQYHNIMTVKRVGIIISCIWAACTVS
GILFIIYSDSSAVIICLITMFFTMLALMASLYVHMFLMARLHIKRIAVLPGTGAIRQGAN
MKGAITLTILIGVFVVCWAPFFLHLIFYISCPQNPYCVCFMSHFNLYLILIMCNSIIDPL
IYALRSQELRKTFKEIICCYPLGGLCDLSSRY
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| BDBM68044 |
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| n/a |
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| Name | BDBM68044 |
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| Synonyms: | 1-(1-naphthalenyloxy)-3-[2-[4-(trifluoromethyl)phenyl]ethylamino]-2-propanol | 1-(1-naphthoxy)-3-[2-[4-(trifluoromethyl)phenyl]ethylamino]propan-2-ol | 1-naphthalen-1-yloxy-3-[2-[4-(trifluoromethyl)phenyl]ethylamino]propan-2-ol | MLS000334371 | SMR000249129 | cid_3605184 |
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| Type | Small organic molecule |
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| Emp. Form. | C22H22F3NO2 |
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| Mol. Mass. | 389.4108 |
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| SMILES | OC(CNCCc1ccc(cc1)C(F)(F)F)COc1cccc2ccccc12 |
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| Structure | 
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