| Reaction Details |
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 | Report a problem with these data |
| Target | Melanocortin receptor 4 |
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| Ligand | BDBM63097 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | TRFRET-based cell-based high throughput dose response assay for biased ligands (antagonists) of the melanocortin 4 receptor (MC4R) |
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| IC50 | >64598±n/a nM |
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| Citation |  PubChem, PC TRFRET-based cell-based high throughput dose response assay for biased ligands (antagonists) of the melanocortin 4 receptor (MC4R) PubChem Bioassay(2012)[AID] |
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| More Info.: | Get all data from this article, Assay Method |
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| Melanocortin receptor 4 |
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| Name: | Melanocortin receptor 4 |
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| Synonyms: | MC4-R | MC4R | MC4R_HUMAN | Melanocortin MC4 | Melanocortin receptor 4 (MC-4) | Melanocortin receptor 4 (MC4-R) | Melanocortin receptor 4 (MC4R) |
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| Type: | Enzyme |
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| Mol. Mass.: | 36949.50 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P32245 |
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| Residue: | 332 |
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| Sequence: | MVNSTHRGMHTSLHLWNRSSYRLHSNASESLGKGYSDGGCYEQLFVSPEVFVTLGVISLL
ENILVIVAIAKNKNLHSPMYFFICSLAVADMLVSVSNGSETIVITLLNSTDTDAQSFTVN
IDNVIDSVICSSLLASICSLLSIAVDRYFTIFYALQYHNIMTVKRVGIIISCIWAACTVS
GILFIIYSDSSAVIICLITMFFTMLALMASLYVHMFLMARLHIKRIAVLPGTGAIRQGAN
MKGAITLTILIGVFVVCWAPFFLHLIFYISCPQNPYCVCFMSHFNLYLILIMCNSIIDPL
IYALRSQELRKTFKEIICCYPLGGLCDLSSRY
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| BDBM63097 |
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| n/a |
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| Name | BDBM63097 |
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| Synonyms: | MLS000556132 | N-[2-(cyclopentylamino)-2-keto-1-(2-thienyl)ethyl]-N-(2,5-dimethoxyphenyl)propiolamide | N-[2-(cyclopentylamino)-2-oxidanylidene-1-thiophen-2-yl-ethyl]-N-(2,5-dimethoxyphenyl)prop-2-ynamide | N-[2-(cyclopentylamino)-2-oxo-1-thiophen-2-ylethyl]-N-(2,5-dimethoxyphenyl)-2-propynamide | N-[2-(cyclopentylamino)-2-oxo-1-thiophen-2-ylethyl]-N-(2,5-dimethoxyphenyl)prop-2-ynamide | Propynoic acid (cyclopentylcarbamoyl-thiophen-2-yl-methyl)-(2,5-dimethoxy-phenyl)-amide | SMR000173283 | cid_3216694 |
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| Type | Small organic molecule |
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| Emp. Form. | C22H24N2O4S |
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| Mol. Mass. | 412.502 |
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| SMILES | COc1ccc(OC)c(c1)N(C(C(=O)NC1CCCC1)c1cccs1)C(=O)C#C |
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| Structure | 
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