| Reaction Details |
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 | Report a problem with these data |
| Target | Dual specificity protein phosphatase 3 |
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| Ligand | BDBM88739 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Dose Response selectivity of inhibitors of STriatal-Enriched Phosphatase (STEP) in the dual-specificity protein-tyrosine phosphatase VHR Inhibition Assay |
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| IC50 | 3400±n/a nM |
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| Citation |  PubChem, PC Dose Response selectivity of inhibitors of STriatal-Enriched Phosphatase (STEP) in the dual-specificity protein-tyrosine phosphatase VHR Inhibition Assay PubChem Bioassay(2012)[AID] |
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| More Info.: | Get all data from this article, Assay Method |
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| |
| Dual specificity protein phosphatase 3 |
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| Name: | Dual specificity protein phosphatase 3 |
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| Synonyms: | DUS3_HUMAN | DUSP3 | Dual specificity protein phosphatase (VHR) | Dual specificity protein phosphatase 3 | Dual specificity protein phosphatase VHR | Protein Tyrosine Phosphatase VHR | Tyrosine-protein phosphatase non-receptor type 1 | VHR |
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| Type: | Hydrolase |
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| Mol. Mass.: | 20480.58 |
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| Organism: | Homo sapiens (Human) |
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| Description: | n/a |
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| Residue: | 185 |
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| Sequence: | MSGSFELSVQDLNDLLSDGSGCYSLPSQPCNEVTPRIYVGNASVAQDIPKLQKLGITHVL
NAAEGRSFMHVNTNANFYKDSGITYLGIKANDTQEFNLSAYFERAADFIDQALAQKNGRV
LVHCREGYSRSPTLVIAYLMMRQKMDVKSALSIVRQNREIGPNDGFLAQLCQLNDRLAKE
GKLKP
|
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|
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| BDBM88739 |
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| n/a |
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| Name | BDBM88739 |
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| Synonyms: | MLS000704210 | N'-[(5-bromo-2-thienyl)methylene]-3-nitrobenzohydrazide | N-[(E)-(5-bromanylthiophen-2-yl)methylideneamino]-3-nitro-benzamide | N-[(E)-(5-bromo-2-thienyl)methyleneamino]-3-nitro-benzamide | N-[(E)-(5-bromo-2-thiophenyl)methylideneamino]-3-nitrobenzamide | N-[(E)-(5-bromothiophen-2-yl)methylideneamino]-3-nitrobenzamide | SMR000227120 | cid_6872971 |
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| Type | Small organic molecule |
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| Emp. Form. | C12H8BrN3O3S |
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| Mol. Mass. | 354.179 |
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| SMILES | [O-][N+](=O)c1cccc(c1)C(=O)N\N=C\c1ccc(Br)s1 |
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| Structure | 
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