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TargetHigh affinity choline transporter 1
LigandBDBM89148
Substrate/Competitorn/a
Meas. Tech.Dose responses of compounds that activate the Choline Transporter (CHT) - 10 point CRC
EC50 24710±n/a nM
Citation PubChem, PC Dose responses of compounds that activate the Choline Transporter (CHT) - 10 point CRC PubChem Bioassay(2012)[AID]
More Info.:Get all data from this article,  Assay Method
 
High affinity choline transporter 1
Name:High affinity choline transporter 1
Synonyms:CHT1 | High-affinity choline transporter | SC5A7_HUMAN | SLC5A7 | high affinity choline transporter 1
Type:PROTEIN
Mol. Mass.:63194.33
Organism:Homo sapiens (Human)
Description:ChEMBL_1464247
Residue:580
Sequence:
MAFHVEGLIAIIVFYLLILLVGIWAAWRTKNSGSAEERSEAIIVGGRDIGLLVGGFTMTA
TWVGGGYINGTAEAVYVPGYGLAWAQAPIGYSLSLILGGLFFAKPMRSKGYVTMLDPFQQ
IYGKRMGGLLFIPALMGEMFWAAAIFSALGATISVIIDVDMHISVIISALIATLYTLVGG
LYSVAYTDVVQLFCIFVGLWISVPFALSHPAVADIGFTAVHAKYQKPWLGTVDSSEVYSW
LDSFLLLMLGGIPWQAYFQRVLSSSSATYAQVLSFLAAFGCLVMAIPAILIGAIGASTDW
NQTAYGLPDPKTTEEADMILPIVLQYLCPVYISFFGLGAVSAAVMSSADSSILSASSMFA
RNIYQLSFRQNASDKEIVWVMRITVFVFGASATAMALLTKTVYGLWYLSSDLVYIVIFPQ
LLCVLFVKGTNTYGAVAGYVSGLFLRITGGEPYLYLQPLIFYPGYYPDDNGIYNQKFPFK
TLAMVTSFLTNICISYLAKYLFESGTLPPKLDVFDAVVARHSEENMDKTILVKNENIKLD
ELALVKPRQSMTLSSTFTNKEAFLDVDSSPEGSGTEDNLQ
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  Blast E-value cutoff:
BDBM89148
n/a
NameBDBM89148
Synonyms:4-[4-(3-chlorophenyl)-1-piperazinyl]-N,N-diethyl-3-pyridinesulfonamide | 4-[4-(3-chlorophenyl)piperazin-1-yl]-N,N-diethyl-pyridine-3-sulfonamide | 4-[4-(3-chlorophenyl)piperazin-1-yl]-N,N-diethylpyridine-3-sulfonamide | 4-[4-(3-chlorophenyl)piperazino]-N,N-diethyl-pyridine-3-sulfonamide | MLS000701226 | SMR000231077 | cid_1214515
TypeSmall organic molecule
Emp. Form.C19H25ClN4O2S
Mol. Mass.408.945
SMILESCCN(CC)S(=O)(=O)c1cnccc1N1CCN(CC1)c1cccc(Cl)c1
Structure
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