| Reaction Details |
|---|
 | Report a problem with these data |
| Target | High affinity choline transporter 1 |
|---|
| Ligand | BDBM89155 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | Dose responses of compounds that activate the Choline Transporter (CHT) - 10 point CRC |
|---|
| EC50 | 8420±n/a nM |
|---|
| Citation |  PubChem, PC Dose responses of compounds that activate the Choline Transporter (CHT) - 10 point CRC PubChem Bioassay(2012)[AID] |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| High affinity choline transporter 1 |
|---|
| Name: | High affinity choline transporter 1 |
|---|
| Synonyms: | CHT1 | High-affinity choline transporter | SC5A7_HUMAN | SLC5A7 | high affinity choline transporter 1 |
|---|
| Type: | PROTEIN |
|---|
| Mol. Mass.: | 63194.33 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | ChEMBL_1464247 |
|---|
| Residue: | 580 |
|---|
| Sequence: | MAFHVEGLIAIIVFYLLILLVGIWAAWRTKNSGSAEERSEAIIVGGRDIGLLVGGFTMTA
TWVGGGYINGTAEAVYVPGYGLAWAQAPIGYSLSLILGGLFFAKPMRSKGYVTMLDPFQQ
IYGKRMGGLLFIPALMGEMFWAAAIFSALGATISVIIDVDMHISVIISALIATLYTLVGG
LYSVAYTDVVQLFCIFVGLWISVPFALSHPAVADIGFTAVHAKYQKPWLGTVDSSEVYSW
LDSFLLLMLGGIPWQAYFQRVLSSSSATYAQVLSFLAAFGCLVMAIPAILIGAIGASTDW
NQTAYGLPDPKTTEEADMILPIVLQYLCPVYISFFGLGAVSAAVMSSADSSILSASSMFA
RNIYQLSFRQNASDKEIVWVMRITVFVFGASATAMALLTKTVYGLWYLSSDLVYIVIFPQ
LLCVLFVKGTNTYGAVAGYVSGLFLRITGGEPYLYLQPLIFYPGYYPDDNGIYNQKFPFK
TLAMVTSFLTNICISYLAKYLFESGTLPPKLDVFDAVVARHSEENMDKTILVKNENIKLD
ELALVKPRQSMTLSSTFTNKEAFLDVDSSPEGSGTEDNLQ
|
|
|
|---|
| BDBM89155 |
|---|
| n/a |
|---|
| Name | BDBM89155 |
|---|
| Synonyms: | 4-(isoxazol-3-ylcarbamoylamino)benzoic acid ethyl ester | 4-[[(3-isoxazolylamino)-oxomethyl]amino]benzoic acid ethyl ester | MLS000679330 | SMR000297739 | cid_6468758 | ethyl 4-(1,2-oxazol-3-ylcarbamoylamino)benzoate | ethyl 4-{[(3-isoxazolylamino)carbonyl]amino}benzoate |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C13H13N3O4 |
|---|
| Mol. Mass. | 275.26 |
|---|
| SMILES | CCOC(=O)c1ccc(NC(=O)Nc2ccon2)cc1 |
|---|
| Structure | 
|
|---|
Search and Browse
