| Reaction Details |
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 | Report a problem with these data |
| Target | High affinity choline transporter 1 |
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| Ligand | BDBM61133 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Dose responses of compounds that activate the Choline Transporter (CHT) - 10 point CRC |
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| EC50 | 7330±n/a nM |
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| Citation |  PubChem, PC Dose responses of compounds that activate the Choline Transporter (CHT) - 10 point CRC PubChem Bioassay(2012)[AID] |
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| More Info.: | Get all data from this article, Assay Method |
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| High affinity choline transporter 1 |
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| Name: | High affinity choline transporter 1 |
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| Synonyms: | CHT1 | High-affinity choline transporter | SC5A7_HUMAN | SLC5A7 | high affinity choline transporter 1 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 63194.33 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_1464247 |
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| Residue: | 580 |
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| Sequence: | MAFHVEGLIAIIVFYLLILLVGIWAAWRTKNSGSAEERSEAIIVGGRDIGLLVGGFTMTA
TWVGGGYINGTAEAVYVPGYGLAWAQAPIGYSLSLILGGLFFAKPMRSKGYVTMLDPFQQ
IYGKRMGGLLFIPALMGEMFWAAAIFSALGATISVIIDVDMHISVIISALIATLYTLVGG
LYSVAYTDVVQLFCIFVGLWISVPFALSHPAVADIGFTAVHAKYQKPWLGTVDSSEVYSW
LDSFLLLMLGGIPWQAYFQRVLSSSSATYAQVLSFLAAFGCLVMAIPAILIGAIGASTDW
NQTAYGLPDPKTTEEADMILPIVLQYLCPVYISFFGLGAVSAAVMSSADSSILSASSMFA
RNIYQLSFRQNASDKEIVWVMRITVFVFGASATAMALLTKTVYGLWYLSSDLVYIVIFPQ
LLCVLFVKGTNTYGAVAGYVSGLFLRITGGEPYLYLQPLIFYPGYYPDDNGIYNQKFPFK
TLAMVTSFLTNICISYLAKYLFESGTLPPKLDVFDAVVARHSEENMDKTILVKNENIKLD
ELALVKPRQSMTLSSTFTNKEAFLDVDSSPEGSGTEDNLQ
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| BDBM61133 |
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| n/a |
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| Name | BDBM61133 |
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| Synonyms: | 5-(4-methylsulfanylphenyl)-N,4-diphenyl-1,3,4-thiadiazol-4-ium-2-amine;chloride | 5-[4-(methylthio)phenyl]-N,4-diphenyl-1,3,4-thiadiazol-4-ium-2-amine;chloride | MLS000948408 | SMR000526827 | [5-[4-(methylthio)phenyl]-4-phenyl-1,3,4-thiadiazol-4-ium-2-yl]-phenyl-amine;chloride | cid_24789686 |
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| Type | Small organic molecule |
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| Emp. Form. | C21H18N3S2 |
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| Mol. Mass. | 376.517 |
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| SMILES | CSc1ccc(cc1)-c1sc(Nc2ccccc2)n[n+]1-c1ccccc1 |
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| Structure | 
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