| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Serum paraoxonase/arylesterase 1 |
|---|
| Ligand | BDBM92333 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | Paraoxonase Activity Assay |
|---|
| pH | 10.5±0 |
|---|
| Temperature | 298.15±0 K |
|---|
| Ki | 11116000±0.0 nM |
|---|
| IC50 | 13010000±0.0 nM |
|---|
| Citation |  Ekinci, D; Beydemir, S Effect of some analgesics on paraoxonase-1 purified from human serum. J Enzyme Inhib Med Chem24:1034-9 (2009) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Solution Info, Assay Method |
|---|
| |
| Serum paraoxonase/arylesterase 1 |
|---|
| Name: | Serum paraoxonase/arylesterase 1 |
|---|
| Synonyms: | A-esterase 1 | Aromatic esterase 1 | K-45 | PON | PON 1 | PON1 | PON1_HUMAN | Paraoxonase (PON1) | Paraoxonase (hPON1) | Paraoxonase 1 (PON1) | Serum aryldialkylphosphatase 1 | Serum paraoxonase 1 (PON1) |
|---|
| Type: | Enzyme |
|---|
| Mol. Mass.: | 39719.73 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | P27169 |
|---|
| Residue: | 355 |
|---|
| Sequence: | MAKLIALTLLGMGLALFRNHQSSYQTRLNALREVQPVELPNCNLVKGIETGSEDLEILPN
GLAFISSGLKYPGIKSFNPNSPGKILLMDLNEEDPTVLELGITGSKFDVSSFNPHGISTF
TDEDNAMYLLVVNHPDAKSTVELFKFQEEEKSLLHLKTIRHKLLPNLNDIVAVGPEHFYG
TNDHYFLDPYLQSWEMYLGLAWSYVVYYSPSEVRVVAEGFDFANGINISPDGKYVYIAEL
LAHKIHVYEKHANWTLTPLKSLDFNTLVDNISVDPETGDLWVGCHPNGMKIFFYDSENPP
ASEVLRIQNILTEEPKVTQVYAENGTVLQGSTVASVYKGKLLIGTVFHKALYCEL
|
|
|
|---|
| BDBM92333 |
|---|
| n/a |
|---|
| Name | BDBM92333 |
|---|
| Synonyms: | Lincomycine |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C18H34N2O6S |
|---|
| Mol. Mass. | 406.537 |
|---|
| SMILES | CCCC1CC(N(C)C1)C(=O)NC(C(C)O)C1OC(SC)C(O)C(O)C1O |
|---|
| Structure | 
|
|---|
Search and Browse
