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TargetNociceptin receptor
LigandBDBM86258
Substrate/Competitorn/a
Ki 1000±n/a nM
CommentsPDSP_1250
Citation Mogil, JSPasternak, GW The molecular and behavioral pharmacology of the orphanin FQ/nociceptin peptide and receptor family. Pharmacol Rev53:381-415 (2001) [PubMed]
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Nociceptin receptor
Name:Nociceptin receptor
Synonyms:K3 opiate receptor | KOR-3 | Kappa-type 3 opioid receptor | Nociceptin receptor | Nociceptin/Orphanin FQ, NOP receptor | OPRX_MOUSE | ORGC | Oor | Oprl | Oprl1 | Orphanin FQ receptor
Type:Enzyme Catalytic Domain
Mol. Mass.:40499.09
Organism:MOUSE
Description:Nociceptin/Orphanin FQ, NOP receptor 0 MOUSE::P35377
Residue:367
Sequence:
MESLFPAPFWEVLYGSHFQGNLSLLNETVPHHLLLNASHSAFLPLGLKVTIVGLYLAVCI
GGLLGNCLVMYVILRHTKMKTATNIYIFNLALADTLVLLTLPFQGTDILLGFWPFGNALC
KTVIAIDYYNMFTSTFTLTAMSVDRYVAICHPIRALDVRTSSKAQAVNVAIWALASVVGV
PVAIMGSAQVEDEEIECLVEIPAPQDYWGPVFAICIFLFSFIIPVLIISVCYSLMIRRLR
GVRLLSGSREKDRNLRRITRLVLVVVAVFVGCWTPVQVFVLVQGLGVQPGSETAVAILRF
CTALGYVNSCLNPILYAFLDENFKACFRKFCCASALHREMQVSDRVRSIAKDVGLGCKTS
ETVPRPA
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  Blast E-value cutoff:
BDBM86258
n/a
NameBDBM86258
Synonyms:CAS_23552-18-3 | Morphine | NSC_5980
TypeSmall organic molecule
Emp. Form.C17H19NO3
Mol. Mass.285.3377
SMILESCN1CCC23C4Oc5c2c(CC1C3C=CC4O)ccc5O |c:16,TLB:13:12:1.2.3:10.9.8|
Structure
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