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| Reaction Details | |||
|---|---|---|---|
 | Report a problem with these data | ||
| Target | Sentrin-specific protease 8 | ||
| Ligand | BDBM42151 | ||
| Substrate/Competitor | n/a | ||
| IC50 | 2980±204 nM | ||
| Citation |  PubChem, PC Dose-response confirmation of uHTS inhibitor hits of Sentrin-Specific Protease 8 using a kinetic assay with Nedd8 Protein Substrate PubChem Bioassay(2012)[AID] | ||
| More Info.: | Get all data from this article | ||
| Sentrin-specific protease 8 | |||
| Name: | Sentrin-specific protease 8 | ||
| Synonyms: | DEN1 | NEDP1 | PRSC2 | SENP8 | SENP8_HUMAN | SUMO/sentrin specific peptidase family member 8 | ||
| Type: | Enzyme Catalytic Domain | ||
| Mol. Mass.: | 24104.52 | ||
| Organism: | Homo sapiens (Human) | ||
| Description: | gi_262118306 | ||
| Residue: | 212 | ||
| Sequence: |
| ||
| BDBM42151 | |||
| n/a | |||
| Name | BDBM42151 | ||
| Synonyms: | (5aR,9aS)-10-oxidanidyl-5-oxidanylidene-5a,6,7,8,9,9a-hexahydroindeno[1,2-b]quinoxalin-5-ium-11-one | (5aR,9aS)-10-oxido-5-oxo-5a,6,7,8,9,9a-hexahydroindeno[1,2-b]quinoxalin-5-ium-11-one | (5aR,9aS)-5-keto-10-oxido-5a,6,7,8,9,9a-hexahydroindeno[1,2-b]quinoxalin-5-ium-11-one | (5aR,9aS)-5a,6,7,8,9,9a-hexahydro-11H-indeno[1,2-b]quinoxalin-11-one 5,10-dioxide | MLS000089701 | SMR000024319 | cid_1886595 | ||
| Type | Small organic molecule | ||
| Emp. Form. | C15H14N2O3 | ||
| Mol. Mass. | 270.2833 | ||
| SMILES | [O-]N1[C@H]2CCCC[C@H]2[N+](=O)C2=C1C(=O)c1ccccc21 |c:11| | ||
| Structure | 
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