| Reaction Details |
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 | Report a problem with these data |
| Target | Corticotropin-releasing factor-binding protein |
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| Ligand | BDBM90508 |
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| Substrate/Competitor | n/a |
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| IC50 | 3740±n/a nM |
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| Citation |  PubChem, PC Dose Response confirmation of uHTS hits for small molecule antagonists of the CRF-binding protein and CRF-R2 receptor complex in 384 well format PubChem Bioassay(2012)[AID] |
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| More Info.: | Get all data from this article |
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| Corticotropin-releasing factor-binding protein |
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| Name: | Corticotropin-releasing factor-binding protein |
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| Synonyms: | CRFBP | CRHBP | CRHBP_HUMAN | corticotropin releasing factor-binding protein |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 36143.95 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P24387 |
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| Residue: | 322 |
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| Sequence: | MSPNFKLQCHFILIFLTALRGESRYLELREAADYDPFLLFSANLKRELAGEQPYRRALRC
LDMLSLQGQFTFTADRPQLHCAAFFISEPEEFITIHYDQVSIDCQGGDFLKVFDGWILKG
EKFPSSQDHPLPSAERYIDFCESGLSRRSIRSSQNVAMIFFRVHEPGNGFTLTIKTDPNL
FPCNVISQTPNGKFTLVVPHQHRNCSFSIIYPVVIKISDLTLGHVNGLQLKKSSAGCEGI
GDFVELLGGTGLDPSKMTPLADLCYPFHGPAQMKVGCDNTVVRMVSSGKHVNRVTFEYRQ
LEPYELENPNGNSIGEFCLSGL
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| BDBM90508 |
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| n/a |
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| Name | BDBM90508 |
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| Synonyms: | 2-(3,5-dimethylanilino)-3,4,5,6-tetrafluoro-benzoic acid | 2-(3,5-dimethylanilino)-3,4,5,6-tetrafluorobenzoic acid | 2-[(3,5-dimethylphenyl)amino]-3,4,5,6-tetrafluorobenzoic acid | 2-[(3,5-dimethylphenyl)amino]-3,4,5,6-tetrakis(fluoranyl)benzoic acid | MLS000689735 | SMR000313339 | cid_4549148 |
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| Type | Small organic molecule |
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| Emp. Form. | C15H11F4NO2 |
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| Mol. Mass. | 313.247 |
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| SMILES | Cc1cc(C)cc(Nc2c(F)c(F)c(F)c(F)c2C(O)=O)c1 |
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| Structure | 
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