Reaction Details |
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Target | Perilipin-5 |
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Ligand | BDBM34677 |
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Substrate/Competitor | n/a |
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IC50 | 2531±n/a nM |
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Citation | PubChem, PC Luminescence-based biochemical high throughput dose response assay for inhibitors of the interaction of the lipase co-activator protein, abhydrolase domain containing 5 (ABHD5) with perilipin-5 (MLDP; PLIN5) PubChem Bioassay(2012)[AID] |
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More Info.: | Get all data from this article |
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Perilipin-5 |
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Name: | Perilipin-5 |
Synonyms: | LSDP5 | OXPAT | PAT-1 | PLIN5 | PLIN5_HUMAN |
Type: | Enzyme Catalytic Domain |
Mol. Mass.: | 50774.20 |
Organism: | Homo sapiens (Human) |
Description: | gi_116292172 |
Residue: | 463 |
Sequence: | MSEEEAAQIPRSSVWEQDQQNVVQRVVALPLVRATCTAVCDVYSAAKDRHPLLGSACRLA
ENCVCGLTTRALDHAQPLLEHLQPQLATMNSLACRGLDKLEEKLPFLQQPSETVVTSAKD
VVASSVTGVVDLARRGRRWSVELKRSVSHAVDVVLEKSEELVDHFLPMTEEELAALAAEA
EGPEVGSVEDQRRQQGYFVRLGSLSARIRHLAYEHSVGKLRQSKHRAQDTLAQLQETLEL
IDHMQCGVTPTAPACPGKVHELWGEWGQRPPESRRRSQAELETLVLSRSLTQELQGTVEA
LESSVRGLPAGAQEKVAEVRRSVDALQTAFADARCFRDVPAAALAEGRGRVAHAHACVDE
LLELVVQAVPLPWLVGPFAPILVERPEPLPDLADLVDEVIGGPDPRWAHLDWPAQQRAWE
AEHRDGSGNGDGDRMGVAGDICEQEPETPSCPVKHTLMPELDF
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BDBM34677 |
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n/a |
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Name | BDBM34677 |
Synonyms: | 3-(4-methylbenzoyl)benzo[g][1]benzofuran-4,5-dione | 3-(4-methylbenzoyl)naphtho[1,2-b]furan-4,5-dione | 3-(4-methylphenyl)carbonylbenzo[g][1]benzofuran-4,5-dione | 3-[(4-methylphenyl)-oxomethyl]benzo[g]benzofuran-4,5-dione | 3-p-toluoylbenzo[g]benzofuran-4,5-quinone | MLS000532156 | SMR000137097 | cid_1736341 |
Type | Small organic molecule |
Emp. Form. | C20H12O4 |
Mol. Mass. | 316.3069 |
SMILES | Cc1ccc(cc1)C(=O)c1coc-2c1C(=O)C(=O)c1ccccc-21 |
Structure |
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