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TargetNuclear receptor subfamily 5 group A member 2
LigandBDBM68466
Substrate/Competitorn/a
IC50 11066±n/a nM
Citation PubChem, PC Luminescence-based cell-based high throughput dose response assay for inverse agonists of the liver receptor homolog-1 (LRH-1; NR5A2) PubChem Bioassay(2013)[AID]
More Info.:Get all data from this article
 
Nuclear receptor subfamily 5 group A member 2
Name:Nuclear receptor subfamily 5 group A member 2
Synonyms:Alpha-1-fetoprotein transcription factor | B1-binding factor | B1F | CPF | CYP7A promoter-binding factor | FTF | Hepatocytic transcription factor | LRH-1 | Liver Receptor Homolog 1 | NR5A2 | NR5A2_HUMAN | Nuclear receptor subfamily 5 group A member 2 | hB1F | nuclear receptor subfamily 5 group A member 2 isoform 2
Type:Nuclear Hormone Receptor
Mol. Mass.:61341.37
Organism:Homo sapiens (Human)
Description:n/a
Residue:541
Sequence:
MSSNSDTGDLQESLKHGLTPIGAGLPDRHGSPIPARGRLVMLPKVETEALGLARSHGEQG
QMPENMQVSQFKMVNYSYDEDLEELCPVCGDKVSGYHYGLLTCESCKGFFKRTVQNNKRY
TCIENQNCQIDKTQRKRCPYCRFQKCLSVGMKLEAVRADRMRGGRNKFGPMYKRDRALKQ
QKKALIRANGLKLEAMSQVIQAMPSDLTISSAIQNIHSASKGLPLNHAALPPTDYDRSPF
VTSPISMTMPPHGSLQGYQTYGHFPSRAIKSEYPDPYTSSPESIMGYSYMDSYQTSSPAS
IPHLILELLKCEPDEPQVQAKIMAYLQQEQANRSKHEKLSTFGLMCKMADQTLFSIVEWA
RSSIFFRELKVDDQMKLLQNCWSELLILDHIYRQVVHGKEGSIFLVTGQQVDYSIIASQA
GATLNNLMSHAQELVAKLRSLQFDQREFVCLKFLVLFSLDVKNLENFQLVEGVQEQVNAA
LLDYTMCNYPQQTEKFGQLLLRLPEIRAISMQAEEYLYYKHLNGDVPYNNLLIEMLHAKR
A
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BDBM68466
n/a
NameBDBM68466
Synonyms:2-[2,5-bis(oxidanylidene)pyrrolidin-1-yl]-N-(4-bromophenyl)ethanamide | MLS000057808 | N-(4-bromophenyl)-2-(2,5-dioxo-1-pyrrolidinyl)acetamide | N-(4-bromophenyl)-2-(2,5-dioxopyrrolidin-1-yl)acetamide | N-(4-bromophenyl)-2-succinimido-acetamide | SMR000063192 | cid_2083990
TypeSmall organic molecule
Emp. Form.C12H11BrN2O3
Mol. Mass.311.131
SMILESBrc1ccc(NC(=O)CN2C(=O)CCC2=O)cc1
Structure
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