Reaction Details |
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Target | Nuclear receptor subfamily 5 group A member 2 |
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Ligand | BDBM95586 |
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Substrate/Competitor | n/a |
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IC50 | >3986±n/a nM |
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Citation | PubChem, PC Luminescence-based cell-based high throughput dose response assay for inverse agonists of the liver receptor homolog-1 (LRH-1; NR5A2) PubChem Bioassay(2013)[AID] |
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More Info.: | Get all data from this article |
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Nuclear receptor subfamily 5 group A member 2 |
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Name: | Nuclear receptor subfamily 5 group A member 2 |
Synonyms: | Alpha-1-fetoprotein transcription factor | B1-binding factor | B1F | CPF | CYP7A promoter-binding factor | FTF | Hepatocytic transcription factor | LRH-1 | Liver Receptor Homolog 1 | NR5A2 | NR5A2_HUMAN | Nuclear receptor subfamily 5 group A member 2 | hB1F | nuclear receptor subfamily 5 group A member 2 isoform 2 |
Type: | Nuclear Hormone Receptor |
Mol. Mass.: | 61341.37 |
Organism: | Homo sapiens (Human) |
Description: | n/a |
Residue: | 541 |
Sequence: | MSSNSDTGDLQESLKHGLTPIGAGLPDRHGSPIPARGRLVMLPKVETEALGLARSHGEQG
QMPENMQVSQFKMVNYSYDEDLEELCPVCGDKVSGYHYGLLTCESCKGFFKRTVQNNKRY
TCIENQNCQIDKTQRKRCPYCRFQKCLSVGMKLEAVRADRMRGGRNKFGPMYKRDRALKQ
QKKALIRANGLKLEAMSQVIQAMPSDLTISSAIQNIHSASKGLPLNHAALPPTDYDRSPF
VTSPISMTMPPHGSLQGYQTYGHFPSRAIKSEYPDPYTSSPESIMGYSYMDSYQTSSPAS
IPHLILELLKCEPDEPQVQAKIMAYLQQEQANRSKHEKLSTFGLMCKMADQTLFSIVEWA
RSSIFFRELKVDDQMKLLQNCWSELLILDHIYRQVVHGKEGSIFLVTGQQVDYSIIASQA
GATLNNLMSHAQELVAKLRSLQFDQREFVCLKFLVLFSLDVKNLENFQLVEGVQEQVNAA
LLDYTMCNYPQQTEKFGQLLLRLPEIRAISMQAEEYLYYKHLNGDVPYNNLLIEMLHAKR
A
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BDBM95586 |
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n/a |
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Name | BDBM95586 |
Synonyms: | 2-(2-keto-7-methyl-4-propyl-chromen-5-yl)oxy-N-(2-pyridyl)acetamide | 2-(7-methyl-2-oxidanylidene-4-propyl-chromen-5-yl)oxy-N-pyridin-2-yl-ethanamide | 2-(7-methyl-2-oxo-4-propylchromen-5-yl)oxy-N-pyridin-2-ylacetamide | 2-[(7-methyl-2-oxo-4-propyl-1-benzopyran-5-yl)oxy]-N-(2-pyridinyl)acetamide | MLS001160382 | SMR000652652 | cid_8034762 |
Type | Small organic molecule |
Emp. Form. | C20H20N2O4 |
Mol. Mass. | 352.3838 |
SMILES | CCCc1cc(=O)oc2cc(C)cc(OCC(=O)Nc3ccccn3)c12 |
Structure |
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