| Reaction Details |
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 | Report a problem with these data |
| Target | Nuclear receptor subfamily 5 group A member 2 |
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| Ligand | BDBM95592 |
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| Substrate/Competitor | n/a |
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| IC50 | 167.85±n/a nM |
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| Citation |  PubChem, PC Luminescence-based cell-based high throughput dose response assay for inverse agonists of the liver receptor homolog-1 (LRH-1; NR5A2) PubChem Bioassay(2013)[AID] |
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| More Info.: | Get all data from this article |
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| Nuclear receptor subfamily 5 group A member 2 |
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| Name: | Nuclear receptor subfamily 5 group A member 2 |
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| Synonyms: | Alpha-1-fetoprotein transcription factor | B1-binding factor | B1F | CPF | CYP7A promoter-binding factor | FTF | Hepatocytic transcription factor | LRH-1 | Liver Receptor Homolog 1 | NR5A2 | NR5A2_HUMAN | Nuclear receptor subfamily 5 group A member 2 | hB1F | nuclear receptor subfamily 5 group A member 2 isoform 2 |
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| Type: | Nuclear Hormone Receptor |
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| Mol. Mass.: | 61341.37 |
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| Organism: | Homo sapiens (Human) |
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| Description: | n/a |
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| Residue: | 541 |
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| Sequence: | MSSNSDTGDLQESLKHGLTPIGAGLPDRHGSPIPARGRLVMLPKVETEALGLARSHGEQG
QMPENMQVSQFKMVNYSYDEDLEELCPVCGDKVSGYHYGLLTCESCKGFFKRTVQNNKRY
TCIENQNCQIDKTQRKRCPYCRFQKCLSVGMKLEAVRADRMRGGRNKFGPMYKRDRALKQ
QKKALIRANGLKLEAMSQVIQAMPSDLTISSAIQNIHSASKGLPLNHAALPPTDYDRSPF
VTSPISMTMPPHGSLQGYQTYGHFPSRAIKSEYPDPYTSSPESIMGYSYMDSYQTSSPAS
IPHLILELLKCEPDEPQVQAKIMAYLQQEQANRSKHEKLSTFGLMCKMADQTLFSIVEWA
RSSIFFRELKVDDQMKLLQNCWSELLILDHIYRQVVHGKEGSIFLVTGQQVDYSIIASQA
GATLNNLMSHAQELVAKLRSLQFDQREFVCLKFLVLFSLDVKNLENFQLVEGVQEQVNAA
LLDYTMCNYPQQTEKFGQLLLRLPEIRAISMQAEEYLYYKHLNGDVPYNNLLIEMLHAKR
A
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| BDBM95592 |
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| n/a |
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| Name | BDBM95592 |
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| Synonyms: | 2-(2-keto-4,7-dimethyl-chromen-5-yl)oxy-N-thiazol-2-yl-acetamide | 2-(4,7-dimethyl-2-oxidanylidene-chromen-5-yl)oxy-N-(1,3-thiazol-2-yl)ethanamide | 2-(4,7-dimethyl-2-oxochromen-5-yl)oxy-N-(1,3-thiazol-2-yl)acetamide | 2-[(4,7-dimethyl-2-oxo-1-benzopyran-5-yl)oxy]-N-(2-thiazolyl)acetamide | MLS001160235 | SMR000652760 | cid_8069390 |
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| Type | Small organic molecule |
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| Emp. Form. | C16H14N2O4S |
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| Mol. Mass. | 330.358 |
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| SMILES | Cc1cc(OCC(=O)Nc2nccs2)c2c(C)cc(=O)oc2c1 |
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| Structure | 
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