BindingDB logo
myBDB logout
Reaction Details
Report a problem with these data
TargetGuanine nucleotide-binding protein subunit alpha-15
LigandBDBM96835
Substrate/Competitorn/a
EC50 22156±n/a nM
Citation PubChem, PC Counterscreen for agonists of the human trace amine associated receptor 1 (TAAR1): Fluorescence-based cell-based high throughput dose response assay to identify nonselective Ga16 agonists PubChem Bioassay(2013)[AID]
More Info.:Get all data from this article
 
Guanine nucleotide-binding protein subunit alpha-15
Name:Guanine nucleotide-binding protein subunit alpha-15
Synonyms:G protein alpha 16 | G-protein subunit alpha-16 | G-protein subunit alpha-16 (G alpha-16) | GNA15 | GNA15_HUMAN | GNA16 | Guanine nucleotide-binding protein subunit alpha-15 [Y147C]
Type:Protein
Mol. Mass.:43577.62
Organism:Homo sapiens (Human)
Description:P30679
Residue:374
Sequence:
MARSLTWRCCPWCLTEDEKAAARVDQEINRILLEQKKQDRGELKLLLLGPGESGKSTFIK
QMRIIHGAGYSEEERKGFRPLVYQNIFVSMRAMIEAMERLQIPFSRPESKHHASLVMSQD
PYKVTTFEKRYAAAMQWLWRDAGIRACYERRREFHLLDSAVYYLSHLERITEEGYVPTAQ
DVLRSRMPTTGINEYCFSVQKTNLRIVDVGGQKSERKKWIHCFENVIALIYLASLSEYDQ
CLEENNQENRMKESLALFGTILELPWFKSTSVILFLNKTDILEEKIPTSHLATYFPSFQG
PKQDAEAAKRFILDMYTRMYTGCVDGPEGSKKGARSRRLFSHYTCATDTQNIRKVFKDVR
DSVLARYLDEINLL
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM96835
n/a
NameBDBM96835
Synonyms:4-(1-amino-2-phenylmethoxyethyl)-N-(6-methoxy-2-pyridinyl)-2-thiazolamine | 4-(1-amino-2-phenylmethoxyethyl)-N-(6-methoxypyridin-2-yl)-1,3-thiazol-2-amine | 4-(1-azanyl-2-phenylmethoxy-ethyl)-N-(6-methoxypyridin-2-yl)-1,3-thiazol-2-amine | MLS003123728 | SMR001291766 | [4-(1-amino-2-benzoxy-ethyl)thiazol-2-yl]-(6-methoxy-2-pyridyl)amine | cid_49786599
TypeSmall organic molecule
Emp. Form.C18H20N4O2S
Mol. Mass.356.442
SMILESCOc1cccc(Nc2nc(cs2)C(N)COCc2ccccc2)n1
Structure
Search PDB for entries with ligand similarity:Similarity to this molecule at least: