| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Nuclear receptor subfamily 0 group B member 1 |
|---|
| Ligand | BDBM97207 |
|---|
| Substrate/Competitor | n/a |
|---|
| IC50 | >833.86±n/a nM |
|---|
| Citation |  PubChem, PC Luminescence-based cell-based high throughput dose response assay for inhibitors of the orphan nuclear receptor subfamily 0, group B, member 1 (DAX1; NR0B1): repression of SF-1 (NR5A1) activated StAR promoter by full-length DAX-1 PubChem Bioassay(2013)[AID] |
|---|
| More Info.: | Get all data from this article |
|---|
| |
| Nuclear receptor subfamily 0 group B member 1 |
|---|
| Name: | Nuclear receptor subfamily 0 group B member 1 |
|---|
| Synonyms: | AHC | DAX1 | NR0B1 | NR0B1_HUMAN |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 51729.22 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | gi_5016090 |
|---|
| Residue: | 470 |
|---|
| Sequence: | MAGENHQWQGSILYNMLMSAKQTRAAPEAPETRLVDQCWGCSCGDEPGVGREGLLGGRNV
ALLYRCCFCGKDHPRQGSILYSMLTSAKQTYAAPKAPEATLGPCWGCSCGSDPGVGRAGL
PGGRPVALLYRCCFCGEDHPRQGSILYSLLTSSKQTHVAPAAPEARPGGAWWDRSYFAQR
PGGKEALPGGRATALLYRCCFCGEDHPQQGSTLYCVPTSTNQAQAAPEERPRAPWWDTSS
GALRPVALKSPQVVCEAASAGLLKTLRFVKYLPCFQVLPLDQQLVLVRNCWASLLMLELA
QDRLQFETVEVSEPSMLQKILTTRRRETGGNEPLPVPTLQHHLAPPAEARKVPSASQVQA
IKCFLSKCWSLNISTKEYAYLKGTVLFNPDVPGLQCVKYIQGLQWGTQQILSEHTRMTHQ
GPHDRFIELNSTLFLLRFINANVIAELFFRPIIGTVSMDDMMLEMLCTKI
|
|
|
|---|
| BDBM97207 |
|---|
| n/a |
|---|
| Name | BDBM97207 |
|---|
| Synonyms: | (Z)-3-[4-[2-cyanoethyl(methyl)amino]phenyl]-2-(2-pyridinyl)-2-propenenitrile | (Z)-3-[4-[2-cyanoethyl(methyl)amino]phenyl]-2-(2-pyridyl)acrylonitrile | (Z)-3-[4-[2-cyanoethyl(methyl)amino]phenyl]-2-pyridin-2-yl-prop-2-enenitrile | (Z)-3-[4-[2-cyanoethyl(methyl)amino]phenyl]-2-pyridin-2-ylprop-2-enenitrile | MLS000392107 | SMR000261058 | cid_6153030 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C18H16N4 |
|---|
| Mol. Mass. | 288.3464 |
|---|
| SMILES | CN(CCC#N)c1ccc(\C=C(/C#N)c2ccccn2)cc1 |
|---|
| Structure | 
|
|---|
Search and Browse
