| Reaction Details |
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 | Report a problem with these data |
| Target | Urokinase plasminogen activator surface receptor |
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| Ligand | BDBM50110015 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Enzyme Assay |
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| Temperature | 297.15±0 K |
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| Ki | 120±0.0 nM |
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| Citation |  Stuerzebecher, J; Steinmetzer, T; Schweinitz, A Urokinase inhibitors, production and use thereof US Patent US8476306 Publication Date 7/2/2013 |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Urokinase plasminogen activator surface receptor |
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| Name: | Urokinase plasminogen activator surface receptor |
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| Synonyms: | CD87 | Plasminogen activator urokinase | Plaur | U-PAR | UPAR | UPAR_RAT | URKR |
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| Type: | Protein |
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| Mol. Mass.: | 35754.96 |
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| Organism: | Rattus norvegicus |
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| Description: | P49616 |
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| Residue: | 328 |
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| Sequence: | MGLLRRRLLLLVVVVTTCVPASQGLRCIQCESNQDCLVEECALGQDLCRTTVLREWEDAE
ELEVVTRGCAHKEKTNRTMSYRMGSVIVSLTETVCATNLCNRPRPGARGRPFPRGRYLEC
ASCTSLDQSCERGREQSLQCRYPTEHCIEVVTLQSTERSVKDEPYTKGCGSLPGCPGTAG
FHSNQTFHFLKCCNFTQCNGGPVLDLQSLPPNGFQCYSCEGNSTFGCSYEETSLIDCRGP
MNQCLEATGLDVLGNRSYTVRGCATASWCQGSHVADSFQTHVNLSISCCNGSGCNRPTGG
APGPGPAHLILIASLLLTLRLWGIPLWT
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| BDBM50110015 |
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| n/a |
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| Name | BDBM50110015 |
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| Synonyms: | CHEMBL158936 | N-(BENZYLSULFONYL)SERYL-N~1~-{4-[AMINO(IMINO)METHYL]BENZYL}GLYCINAMIDE | N-[(4-Carbamimidoyl-benzylcarbamoyl)-methyl]-3-hydroxy-2-phenylmethanesulfonylamino-propionamide | US8476306, 6.1 | US8476306, 6.2 |
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| Type | Small organic molecule |
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| Emp. Form. | C20H25N5O5S |
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| Mol. Mass. | 447.508 |
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| SMILES | NC(=N)c1ccc(CNC(=O)CNC(=O)[C@@H](CO)NS(=O)(=O)Cc2ccccc2)cc1 |
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| Structure | 
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