| Reaction Details |
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 | Report a problem with these data |
| Target | Adenosine receptor A1 |
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| Ligand | BDBM99194 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Binding Assay |
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| Ki | 29±0.0 nM |
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| Citation |  Jagtap, P Adenosine compounds and their use thereof US Patent US8501708 Publication Date 8/6/2013 |
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| More Info.: | Get all data from this article, Assay Method |
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| Adenosine receptor A1 |
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| Name: | Adenosine receptor A1 |
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| Synonyms: | AA1R_RABIT | ADENOSINE A1 | ADENOSINE A1 high | ADENOSINE A1 low | ADORA1 | Adenosine receptor A1 (A1) |
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| Type: | Enzyme |
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| Mol. Mass.: | 36566.33 |
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| Organism: | Oryctolagus cuniculus (Rabbit) |
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| Description: | P34970 |
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| Residue: | 328 |
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| Sequence: | MPPSISAFQAAYIGIEVLIALVSVPGNVLVIWAVKVNQALRDATFCFIVSLAVADVAVGA
LVIPLAILINIGPETYFHTCLMVACPVLILTQSSILALLAIAVDRYLRVKIPLRYKAVVT
PRRAAVAIAGCWILSLVVGLTPMFGWNNLREVQRAWAANGSVGEPVIKCEFEKVISMEYM
VYFNFFVWVLPPLLLMVLIYLEVFYLIRRQLSKKASASSGDPHKYYGKELKIAKSLALIL
FLFALSWLPLHILNCVTLFCPSCQKPSILVYTAIFLTHGNSAMNPIVYAFRIHKFRVTFL
KIWNDHFRCRPAPAGDGDEDLPEEKPND
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| BDBM99194 |
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| n/a |
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| Name | BDBM99194 |
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| Synonyms: | US8501708, 14 | US8501708, 15 |
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| Type | Small organic molecule |
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| Emp. Form. | C23H29N5O5 |
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| Mol. Mass. | 455.5069 |
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| SMILES | OC[C@H]1OC([C@H](O)[C@@H]1O)n1cnc2c(NC3CCCCC3OCc3ccccc3)ncnc12 |r| |
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| Structure | 
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