| Reaction Details |
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 | Report a problem with these data |
| Target | Adenosine receptor A3 |
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| Ligand | BDBM99198 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Binding Assay |
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| Ki | 1570±0.0 nM |
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| Citation |  Jagtap, P Adenosine compounds and their use thereof US Patent US8501708 Publication Date 8/6/2013 |
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| More Info.: | Get all data from this article, Assay Method |
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| Adenosine receptor A3 |
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| Name: | Adenosine receptor A3 |
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| Synonyms: | AA3R_RABIT | ADENOSINE A3 | ADORA3 |
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| Type: | Protein |
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| Mol. Mass.: | 36319.35 |
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| Organism: | Oryctolagus cuniculus (rabbit) |
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| Description: | O02667 |
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| Residue: | 319 |
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| Sequence: | MPDNSTTLFLAIRASYIVFEIVIGVCAVVGNVLVIWVIKLNPSLKTTTFYFIFSLALADI
AVGFLVMPLAIVISLGITIGFYSCLVMSCLLLVFTHASIMSLLAIAVDRYLRVKLTVRYR
RVTTQRRIWLALGLCWVVSLLVGFTPMFGWNMKPTLESARNYSDFQCKFDSVIPMEYMVF
FSFFTWILIPLLLMCALYVYIFYIIRNKLVQSFSSFKETGAFYRREFKTAKSLFLVLALF
AGCWLPLSIINCVTYFKCKVPDVVLLVGILLSHANSMMNPIVYACKIQKFKETYLLIFKA
RVTCQPSDSLDPSSEQNSE
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| BDBM99198 |
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| n/a |
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| Name | BDBM99198 |
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| Synonyms: | US8501708, 18 |
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| Type | Small organic molecule |
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| Emp. Form. | C22H26FN5O5 |
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| Mol. Mass. | 459.4707 |
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| SMILES | OC[C@H]1OC([C@H](O)[C@@H]1O)n1cnc2c(NC3CCC[C@@H]3OCc3cccc(F)c3)ncnc12 |r| |
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| Structure | 
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