| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Kallikrein-7 |
|---|
| Ligand | BDBM100058 |
|---|
| Substrate/Competitor | n/a |
|---|
| EC50 | >7723±n/a nM |
|---|
| Citation |  PubChem, PC Fluorescence Intensity-based biochemical primary high throughput dose response assay to identify activators of kallikrein-7 (K7) zymogen PubChem Bioassay(2013)[AID] |
|---|
| More Info.: | Get all data from this article |
|---|
| |
| Kallikrein-7 |
|---|
| Name: | Kallikrein-7 |
|---|
| Synonyms: | KLK7 | KLK7_HUMAN | Kallikrein 7 | Kallikrein-7 | PRSS6 | SCCE | Serine protease 6 | Stratum corneum chymotryptic enzyme | hK7 | hSCCE | kallikrein-7 isoform 1 preproprotein |
|---|
| Type: | PROTEIN |
|---|
| Mol. Mass.: | 27535.05 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | ChEMBL_1469257 |
|---|
| Residue: | 253 |
|---|
| Sequence: | MARSLLLPLQILLLSLALETAGEEAQGDKIIDGAPCARGSHPWQVALLSGNQLHCGGVLV
NERWVLTAAHCKMNEYTVHLGSDTLGDRRAQRIKASKSFRHPGYSTQTHVNDLMLVKLNS
QARLSSMVKKVRLPSRCEPPGTTCTVSGWGTTTSPDVTFPSDLMCVDVKLISPQDCTKVY
KDLLENSMLCAGIPDSKKNACNGDSGGPLVCRGTLQGLVSWGTFPCGQPNDPGVYTQVCK
FTKWINDTMKKHR
|
|
|
|---|
| BDBM100058 |
|---|
| n/a |
|---|
| Name | BDBM100058 |
|---|
| Synonyms: | MLS000718244 | N-cyclopentyl-2-(4-fluorophenyl)-3-imidazo[1,2-a]pyrazinamine | N-cyclopentyl-2-(4-fluorophenyl)imidazo[1,2-a]pyrazin-3-amine | SMR000290512 | cid_4114964 | cyclopentyl-[2-(4-fluorophenyl)imidazo[1,2-a]pyrazin-3-yl]amine |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C17H17FN4 |
|---|
| Mol. Mass. | 296.3421 |
|---|
| SMILES | Fc1ccc(cc1)-c1nc2cnccn2c1NC1CCCC1 |
|---|
| Structure | 
|
|---|
Search and Browse
