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TargetKallikrein-7
LigandBDBM100070
Substrate/Competitorn/a
EC50 6338±n/a nM
Citation PubChem, PC Fluorescence Intensity-based biochemical primary high throughput dose response assay to identify activators of kallikrein-7 (K7) zymogen PubChem Bioassay(2013)[AID]
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Kallikrein-7
Name:Kallikrein-7
Synonyms:KLK7 | KLK7_HUMAN | Kallikrein 7 | Kallikrein-7 | PRSS6 | SCCE | Serine protease 6 | Stratum corneum chymotryptic enzyme | hK7 | hSCCE | kallikrein-7 isoform 1 preproprotein
Type:PROTEIN
Mol. Mass.:27535.05
Organism:Homo sapiens (Human)
Description:ChEMBL_1469257
Residue:253
Sequence:
MARSLLLPLQILLLSLALETAGEEAQGDKIIDGAPCARGSHPWQVALLSGNQLHCGGVLV
NERWVLTAAHCKMNEYTVHLGSDTLGDRRAQRIKASKSFRHPGYSTQTHVNDLMLVKLNS
QARLSSMVKKVRLPSRCEPPGTTCTVSGWGTTTSPDVTFPSDLMCVDVKLISPQDCTKVY
KDLLENSMLCAGIPDSKKNACNGDSGGPLVCRGTLQGLVSWGTFPCGQPNDPGVYTQVCK
FTKWINDTMKKHR
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BDBM100070
n/a
NameBDBM100070
Synonyms:7-(diethylamino)-3-(hydroxymethyl)-4-methyl-1-benzopyran-2-one | 7-(diethylamino)-3-(hydroxymethyl)-4-methyl-2H-chromen-2-one | 7-(diethylamino)-3-(hydroxymethyl)-4-methyl-chromen-2-one | 7-(diethylamino)-3-(hydroxymethyl)-4-methylchromen-2-one | 7-(diethylamino)-4-methyl-3-methylol-coumarin | MLS000766701 | SMR000339597 | cid_747166
TypeSmall organic molecule
Emp. Form.C15H19NO3
Mol. Mass.261.3163
SMILESCCN(CC)c1ccc2c(C)c(CO)c(=O)oc2c1
Structure
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