| Reaction Details |
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 | Report a problem with these data |
| Target | COUP transcription factor 2 |
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| Ligand | BDBM36871 |
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| Substrate/Competitor | n/a |
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| IC50 | 3111±n/a nM |
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| Citation |  PubChem, PC Luminescence-based cell-based high throughput dose response assay to identify inhibitors of COUP-TFII (NR2F2) PubChem Bioassay(2013)[AID] |
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| More Info.: | Get all data from this article |
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| COUP transcription factor 2 |
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| Name: | COUP transcription factor 2 |
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| Synonyms: | ARP1 | COT2_HUMAN | COUP transcription factor 2 isoform a | NR2F2 | TFCOUP2 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 45583.83 |
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| Organism: | Homo sapiens (Human) |
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| Description: | gi_14149746 |
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| Residue: | 414 |
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| Sequence: | MAMVVSTWRDPQDEVPGSQGSQASQAPPVPGPPPGAPHTPQTPGQGGPASTPAQTAAGGQ
GGPGGPGSDKQQQQQHIECVVCGDKSSGKHYGQFTCEGCKSFFKRSVRRNLSYTCRANRN
CPIDQHHRNQCQYCRLKKCLKVGMRREAVQRGRMPPTQPTHGQFALTNGDPLNCHSYLSG
YISLLLRAEPYPTSRFGSQCMQPNNIMGIENICELAARMLFSAVEWARNIPFFPDLQITD
QVALLRLTWSELFVLNAAQCSMPLHVAPLLAAAGLHASPMSADRVVAFMDHIRIFQEQVE
KLKALHVDSAEYSCLKAIVLFTSDACGLSDVAHVESLQEKSQCALEEYVRSQYPNQPTRF
GKLLLRLPSLRTVSSSVIEQLFFVRLVGKTPIETLIRDMLLSGSSFNWPYMAIQ
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| BDBM36871 |
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| n/a |
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| Name | BDBM36871 |
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| Synonyms: | MLS000027766 | N-[4-(1-Methanesulfonyl-2-methyl-2,3-dihydro-1H-indol-5-yl)-thiazol-2-yl]-2-thiophen-2-yl-acetamide | N-[4-(1-mesyl-2-methyl-indolin-5-yl)thiazol-2-yl]-2-(2-thienyl)acetamide | N-[4-(2-methyl-1-methylsulfonyl-2,3-dihydroindol-5-yl)-1,3-thiazol-2-yl]-2-thiophen-2-yl-ethanamide | N-[4-(2-methyl-1-methylsulfonyl-2,3-dihydroindol-5-yl)-1,3-thiazol-2-yl]-2-thiophen-2-ylacetamide | N-[4-(2-methyl-1-methylsulfonyl-2,3-dihydroindol-5-yl)-2-thiazolyl]-2-thiophen-2-ylacetamide | SMR000007522 | cid_654842 |
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| Type | Small organic molecule |
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| Emp. Form. | C19H19N3O3S3 |
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| Mol. Mass. | 433.567 |
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| SMILES | CC1Cc2cc(ccc2N1S(C)(=O)=O)-c1csc(NC(=O)Cc2cccs2)n1 |
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| Structure | 
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