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| Reaction Details | |||
|---|---|---|---|
 | Report a problem with these data | ||
| Target | Carboxypeptidase B2 | ||
| Ligand | BDBM109240 | ||
| Substrate/Competitor | n/a | ||
| Meas. Tech. | Enzyme Inhibition Assay | ||
| IC50 | 14±n/a nM | ||
| Citation |  Nagata, T; Inoue, M; Ashida, Y; Noguchi, K; Ono, M Cycloalkyl-substituted imidazole derivative US Patent US8609710 Publication Date 12/17/2013 | ||
| More Info.: | Get all data from this article, Assay Method | ||
| Carboxypeptidase B2 | |||
| Name: | Carboxypeptidase B2 | ||
| Synonyms: | CBPB2_HUMAN | CPB2 | CPU | Carboxypeptidase B2 | Carboxypeptidase B2 isoform A | Carboxypeptidase U | Plasma carboxypeptidase B | TAFI | Thrombin-activable fibrinolysis inhibitor | pCPB | ||
| Type: | Enzyme | ||
| Mol. Mass.: | 48432.74 | ||
| Organism: | Homo sapiens (Human) | ||
| Description: | Q96IY4 | ||
| Residue: | 423 | ||
| Sequence: |
| ||
| BDBM109240 | |||
| n/a | |||
| Name | BDBM109240 | ||
| Synonyms: | US8609710, 4 | ||
| Type | Small organic molecule | ||
| Emp. Form. | C15H25N3O2 | ||
| Mol. Mass. | 279.3779 | ||
| SMILES | CCC1CC(C1)n1cnc(CC(CCCN)C(O)=O)c1 |(-4.82,4.9,;-3.34,4.5,;-2.94,3.02,;-1.6,2.25,;-2.37,.91,;-3.71,1.68,;-1.98,-.58,;-2.88,-1.82,;-1.98,-3.07,;-.51,-2.59,;.82,-3.36,;2.16,-2.59,;2.16,-1.05,;3.49,-.28,;3.49,1.26,;4.82,2.03,;3.49,-3.36,;3.49,-4.9,;4.82,-2.59,;-.51,-1.05,)| | ||
| Structure | 
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