| Reaction Details |
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 | Report a problem with these data |
| Target | 5-hydroxytryptamine receptor 2A |
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| Ligand | BDBM114613 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Late stage for the probe development effort to identify agonists of the mouse 5-hydroxytryptamine (serotonin) receptor 2A (HTR2A) |
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| EC50 | 76083±n/a nM |
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| Citation |  PubChem, PC Late stage for the probe development effort to identify agonists of the mouse 5-hydroxytryptamine (serotonin) receptor 2A (HTR2A): Luminescence-based cell-based high throughput dose response assay for agonists of the mouse 5-hydroxytryptamine (serotonin) receptor 2A (HTR2A) PubChem Bioassay(2013)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| 5-hydroxytryptamine receptor 2A |
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| Name: | 5-hydroxytryptamine receptor 2A |
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| Synonyms: | 5-HT-2 | 5-HT-2A | 5-hydroxytryptamine receptor 2A | 5-hydroxytryptamine receptor 2A (5HT2A) | 5HT2A_MOUSE | Dopamine D2 receptor/Serotonin 2 (5-HT2) receptor | Htr2 | Htr2a | Serotonin 2a (5-HT2a) receptor |
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| Type: | Enzyme |
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| Mol. Mass.: | 52843.00 |
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| Organism: | Mus musculus (Mouse) |
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| Description: | P35363 |
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| Residue: | 471 |
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| Sequence: | MEILCEDNISLSSIPNSLMQLGDDSRLYPNDFNSRDANTSEASNWTIDAENRTNLSCEGY
LPPTCLSILHLQEKNWSALLTTVVIILTIAGNILVIMAVSLEKKLQNATNYFLMSLAIAD
MLLGFLVMPVSMLTILYGYRWPLPSKLCAVWIYLDVLFSTASIMHLCAISLDRYVAIQNP
IHHSRFNSRTKAFLKIIAVWTISVGISMPIPVFGLQDDSKVFKEGSCLLADDNFVLIGSF
VAFFIPLTIMVITYFLTIKSLQKEATLCVSDLSTRAKLSSFSFLPQSSLSSEKLFQRSIH
REPGSYAGRRTMQSISNEQKACKVLGIVFFLFVVMWCPFFITNIMAVICKESCNENVIGA
LLNVFVWIGYLSSAVNPLVYTLFNKTYRSAFSRYIQCQYKENRKPLQLILVNTIPTLAYK
SSQLQVGQKKNSQEDAEPTANDCSMVTLGNQHSEEMCTDNIETVNEKVSCV
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| BDBM114613 |
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| n/a |
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| Name | BDBM114613 |
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| Synonyms: | 1-[(5-bromanylthiophen-2-yl)methyl]-4-pyridin-2-yl-piperazine | 1-[(5-bromo-2-thienyl)methyl]-4-(2-pyridyl)piperazine | 1-[(5-bromo-2-thiophenyl)methyl]-4-(2-pyridinyl)piperazine | 1-[(5-bromothiophen-2-yl)methyl]-4-pyridin-2-ylpiperazine | SR-01000202086 | SR-01000202086-3 | cid_2838302 |
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| Type | Small organic molecule |
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| Emp. Form. | C14H16BrN3S |
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| Mol. Mass. | 338.266 |
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| SMILES | Brc1ccc(CN2CCN(CC2)c2ccccn2)s1 |
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| Structure | 
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