| Reaction Details |
|---|
 | Report a problem with these data |
| Target | 5-hydroxytryptamine receptor 2A |
|---|
| Ligand | BDBM114622 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | Late stage for the probe development effort to identify agonists of the mouse 5-hydroxytryptamine (serotonin) receptor 2A (HTR2A) |
|---|
| EC50 | 76083±n/a nM |
|---|
| Citation |  PubChem, PC Late stage for the probe development effort to identify agonists of the mouse 5-hydroxytryptamine (serotonin) receptor 2A (HTR2A): Luminescence-based cell-based high throughput dose response assay for agonists of the mouse 5-hydroxytryptamine (serotonin) receptor 2A (HTR2A) PubChem Bioassay(2013)[AID] |
|---|
| More Info.: | Get all data from this article, Solution Info, Assay Method |
|---|
| |
| 5-hydroxytryptamine receptor 2A |
|---|
| Name: | 5-hydroxytryptamine receptor 2A |
|---|
| Synonyms: | 5-HT-2 | 5-HT-2A | 5-hydroxytryptamine receptor 2A | 5-hydroxytryptamine receptor 2A (5HT2A) | 5HT2A_MOUSE | Dopamine D2 receptor/Serotonin 2 (5-HT2) receptor | Htr2 | Htr2a | Serotonin 2a (5-HT2a) receptor |
|---|
| Type: | Enzyme |
|---|
| Mol. Mass.: | 52843.00 |
|---|
| Organism: | Mus musculus (Mouse) |
|---|
| Description: | P35363 |
|---|
| Residue: | 471 |
|---|
| Sequence: | MEILCEDNISLSSIPNSLMQLGDDSRLYPNDFNSRDANTSEASNWTIDAENRTNLSCEGY
LPPTCLSILHLQEKNWSALLTTVVIILTIAGNILVIMAVSLEKKLQNATNYFLMSLAIAD
MLLGFLVMPVSMLTILYGYRWPLPSKLCAVWIYLDVLFSTASIMHLCAISLDRYVAIQNP
IHHSRFNSRTKAFLKIIAVWTISVGISMPIPVFGLQDDSKVFKEGSCLLADDNFVLIGSF
VAFFIPLTIMVITYFLTIKSLQKEATLCVSDLSTRAKLSSFSFLPQSSLSSEKLFQRSIH
REPGSYAGRRTMQSISNEQKACKVLGIVFFLFVVMWCPFFITNIMAVICKESCNENVIGA
LLNVFVWIGYLSSAVNPLVYTLFNKTYRSAFSRYIQCQYKENRKPLQLILVNTIPTLAYK
SSQLQVGQKKNSQEDAEPTANDCSMVTLGNQHSEEMCTDNIETVNEKVSCV
|
|
|
|---|
| BDBM114622 |
|---|
| n/a |
|---|
| Name | BDBM114622 |
|---|
| Synonyms: | 2-[4-(2,4-dimethylbenzyl)piperazino]pyrimidine | 2-[4-[(2,4-dimethylphenyl)methyl]-1-piperazinyl]pyrimidine | 2-[4-[(2,4-dimethylphenyl)methyl]piperazin-1-yl]pyrimidine | SR-01000201709 | SR-01000201709-3 | cid_763322 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C17H22N4 |
|---|
| Mol. Mass. | 282.3834 |
|---|
| SMILES | Cc1ccc(CN2CCN(CC2)c2ncccn2)c(C)c1 |
|---|
| Structure | 
|
|---|
Search and Browse
