| Reaction Details |
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 | Report a problem with these data |
| Target | PC4 and SFRS1-interacting protein |
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| Ligand | BDBM115127 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Counterscreen for inhibitors of LEDGF/p75-dependent integration: TR-FRET-based biochemical high throughput dose response counterscreen assay to identify activators of HIV-1 Integrase multimerization |
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| IC50 | 4190±n/a nM |
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| Citation |  PubChem, PC Counterscreen for inhibitors of LEDGF/p75-dependent integration: TR-FRET-based biochemical high throughput dose response counterscreen assay to identify activators of HIV-1 Integrase multimerization PubChem Bioassay(2014)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| PC4 and SFRS1-interacting protein |
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| Name: | PC4 and SFRS1-interacting protein |
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| Synonyms: | DFS70 | LEDGF | LEDGF/p75 | PSIP1 | PSIP1_HUMAN | PSIP2 | lens epithelium-derived growth factor p75 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 60120.68 |
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| Organism: | Homo sapiens (Human) |
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| Description: | gi_6708281 |
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| Residue: | 530 |
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| Sequence: | MTRDFKPGDLIFAKMKGYPHWPARVDEVPDGAVKPPTNKLPIFFFGTHETAFLGPKDIFP
YSENKEKYGKPNKRKGFNEGLWEIDNNPKVKFSSQQAATKQSNASSDVEVEEKETSVSKE
DTDHEEKASNEDVTKAVDITTPKAARRGRKRKAEKQVETEEAGVVTTATASVNLKVSPKR
GRPAATEVKIPKPRGRPKMVKQPCPSESDIITEEDKSKKKGQEEKQPKKQPKKDEEGQKE
EDKPRKEPDKKEGKKEVESKRKNLAKTGVTSTSDSEEEGDDQEGEKKRKGGRNFQTAHRR
NMLKGQHEKEAADRKRKQEEQMETEQQNKDEGKKPEVKKVEKKRETSMDSRLQRIHAEIK
NSLKIDNLDVNRCIEALDELASLQVTMQQAQKHTEMITTLKKIRRFKVSQVIMEKSTMLY
NKFKNMFLVGEGDSVITQVLNKSLAEQRQHEEANKTKDQGKKGPNKKLEKEQTGSKTLNG
GSDAQDGNQPQHNGESNEDSKDNHEASTKKKPSSEERETEISLKDSTLDN
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| BDBM115127 |
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| n/a |
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| Name | BDBM115127 |
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| Synonyms: | 4,5,7-trihydroxy-9,10-diketo-anthracene-2-carboxylic acid | 4,5,7-trihydroxy-9,10-dioxo-2-anthracenecarboxylic acid | 4,5,7-trihydroxy-9,10-dioxoanthracene-2-carboxylic acid | 4,5,7-tris(oxidanyl)-9,10-bis(oxidanylidene)anthracene-2-carboxylic acid | MLS000876948 | SMR000440655 | cid_361510 |
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| Type | Small organic molecule |
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| Emp. Form. | C15H8O7 |
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| Mol. Mass. | 300.2198 |
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| SMILES | OC(=O)c1cc(O)c2C(=O)c3c(O)cc(O)cc3C(=O)c2c1 |
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| Structure | 
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