| Reaction Details |
|---|
 | Report a problem with these data |
| Target | PC4 and SFRS1-interacting protein |
|---|
| Ligand | BDBM115152 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | Counterscreen for inhibitors of LEDGF/p75-dependent integration: TR-FRET-based biochemical high throughput dose response counterscreen assay to identify activators of HIV-1 Integrase multimerization |
|---|
| IC50 | 1989±n/a nM |
|---|
| Citation |  PubChem, PC Counterscreen for inhibitors of LEDGF/p75-dependent integration: TR-FRET-based biochemical high throughput dose response counterscreen assay to identify activators of HIV-1 Integrase multimerization PubChem Bioassay(2014)[AID] |
|---|
| More Info.: | Get all data from this article, Solution Info, Assay Method |
|---|
| |
| PC4 and SFRS1-interacting protein |
|---|
| Name: | PC4 and SFRS1-interacting protein |
|---|
| Synonyms: | DFS70 | LEDGF | LEDGF/p75 | PSIP1 | PSIP1_HUMAN | PSIP2 | lens epithelium-derived growth factor p75 |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 60120.68 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | gi_6708281 |
|---|
| Residue: | 530 |
|---|
| Sequence: | MTRDFKPGDLIFAKMKGYPHWPARVDEVPDGAVKPPTNKLPIFFFGTHETAFLGPKDIFP
YSENKEKYGKPNKRKGFNEGLWEIDNNPKVKFSSQQAATKQSNASSDVEVEEKETSVSKE
DTDHEEKASNEDVTKAVDITTPKAARRGRKRKAEKQVETEEAGVVTTATASVNLKVSPKR
GRPAATEVKIPKPRGRPKMVKQPCPSESDIITEEDKSKKKGQEEKQPKKQPKKDEEGQKE
EDKPRKEPDKKEGKKEVESKRKNLAKTGVTSTSDSEEEGDDQEGEKKRKGGRNFQTAHRR
NMLKGQHEKEAADRKRKQEEQMETEQQNKDEGKKPEVKKVEKKRETSMDSRLQRIHAEIK
NSLKIDNLDVNRCIEALDELASLQVTMQQAQKHTEMITTLKKIRRFKVSQVIMEKSTMLY
NKFKNMFLVGEGDSVITQVLNKSLAEQRQHEEANKTKDQGKKGPNKKLEKEQTGSKTLNG
GSDAQDGNQPQHNGESNEDSKDNHEASTKKKPSSEERETEISLKDSTLDN
|
|
|
|---|
| BDBM115152 |
|---|
| n/a |
|---|
| Name | BDBM115152 |
|---|
| Synonyms: | 2-methyl-2-propenoic acid [4-(4-methylphenyl)azo-7-oxo-1-cyclohepta-1,3,5-trienyl] ester | 2-methylacrylic acid [7-keto-4-(p-tolylazo)cyclohepta-1,3,5-trien-1-yl] ester | MLS002694133 | SMR001560064 | [4-[(4-methylphenyl)diazenyl]-7-oxidanylidene-cyclohepta-1,3,5-trien-1-yl] 2-methylprop-2-enoate | [4-[(4-methylphenyl)diazenyl]-7-oxocyclohepta-1,3,5-trien-1-yl] 2-methylprop-2-enoate | cid_254859 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C18H16N2O3 |
|---|
| Mol. Mass. | 308.3312 |
|---|
| SMILES | CC(=C)C(=O)Oc1ccc(ccc1=O)\N=N\c1ccc(C)cc1 |
|---|
| Structure | 
|
|---|
Search and Browse
