| Reaction Details |
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 | Report a problem with these data |
| Target | Egl nine homolog 1 |
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| Ligand | BDBM123039 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Enzyme Assay |
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| Temperature | 298.15±n/a K |
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| IC50 | 30±n/a nM |
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| Comments | extracted |
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| Citation |  Kang, X; Long, W; Ma, C; Wang, Y; Cao, H; Wang, Y; Tan, F; Hu, Y Compounds as hypoxia mimetics, and compositions and uses thereof US Patent US8742138 Publication Date 6/3/2014 |
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| More Info.: | Get all data from this article, Assay Method |
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| Egl nine homolog 1 |
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| Name: | Egl nine homolog 1 |
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| Synonyms: | EGLN1_RAT | Egln1 | Hypoxia-inducible factor (HIF-PH2) |
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| Type: | Enzyme |
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| Mol. Mass.: | 36098.74 |
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| Organism: | Rattus norvegicus (Rat) |
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| Description: | P59722 |
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| Residue: | 338 |
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| Sequence: | PRAQPAPAQPRVAPPPGGAPGAARAGGAARRGDSSTAASRVPGPEDATQAGSGPGPAEPS
SEDPPPSRSPGPERASLCPAGGGPGEALSPSGGLRPNGQTKPLPALKLALEYIVPCMNKH
GICVVDDFLGRETGQQIGDEVRALHDTGKFTDGQLVSQKSDSSKDIRGDKITWIEGKEPG
CETIGLLMSSMDDLIRHCSGKLGNYRINGRTKAMVACYPGNGTGYVRHVDNPNGDGRCVT
CIYYLNKDWDAKVSGGILRIFPEGKAQFADIEPKFDRLLFFWSDRRNPHEVQPAYATRYA
ITVWYFDADERARAKVKYLTGEKGVRVELKPNSVSKDV
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| BDBM123039 |
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| n/a |
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| Name | BDBM123039 |
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| Synonyms: | US8742138, 24 |
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| Type | Small organic molecule |
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| Emp. Form. | C18H11Cl2NO6 |
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| Mol. Mass. | 408.189 |
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| SMILES | OC(=O)CNC(=O)c1c2c(cccc2c(O)oc1=O)-c1ccc(Cl)c(Cl)c1 |
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| Structure | 
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