| Reaction Details |
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 | Report a problem with these data |
| Target | Calcitonin gene-related peptide 1 |
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| Ligand | BDBM126174 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Binding Assay |
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| pH | 7.4±n/a |
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| Temperature | 298.15±n/a K |
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| Ki | 6.6±n/a nM |
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| Comments | extracted |
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| Citation |  Stump, CA; Quigley, AG CGRP receptor antagonists US Patent US8778957 Publication Date 7/15/2014 |
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| More Info.: | Get all data from this article, Assay Method |
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| |
| Calcitonin gene-related peptide 1 |
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| Name: | Calcitonin gene-related peptide 1 |
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| Synonyms: | CALC1 | CALCA | CALCA_HUMAN | CGRP | Calcitonin gene-related peptide (CGRP alpha) | Calcitonin gene-related peptide 1 |
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| Type: | Enzyme |
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| Mol. Mass.: | 13902.80 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P06881 |
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| Residue: | 128 |
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| Sequence: | MGFQKFSPFLALSILVLLQAGSLHAAPFRSALESSPADPATLSEDEARLLLAALVQDYVQ
MKASELEQEQEREGSRIIAQKRACDTATCVTHRLAGLLSRSGGVVKNNFVPTNVGSKAFG
RRRRDLQA
|
|
|
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| BDBM126174 |
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| n/a |
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| Name | BDBM126174 |
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| Synonyms: | US8778957, 64 |
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| Type | Small organic molecule |
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| Emp. Form. | C29H27N5O |
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| Mol. Mass. | 461.5576 |
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| SMILES | O=C1Nc2ncccc2[C@@]11Cc2cc3ccc(CN4CCNCC4c4ccccc4)nc3cc2C1 |r| |
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| Structure | 
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