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Reaction Details
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TargetTransthyretin
LigandBDBM50308499
Substrate/Competitorn/a
Meas. Tech.Luminescence-based cell-based high throughput dose response assay to identify activators of Transthyretin (TTR) transcription
EC50>167158±n/a nM
Citation PubChem, PC Luminescence-based cell-based high throughput dose response assay to identify activators of Transthyretin (TTR) transcription PubChem Bioassay(2014)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Transthyretin
Name:Transthyretin
Synonyms:ATTR | PALB | Prealbumin | TBPA | TTHY_HUMAN | TTR | Transthyretin (TTR)
Type:Enzyme
Mol. Mass.:15884.31
Organism:Homo sapiens (Human)
Description:P02766
Residue:147
Sequence:
MASHRLLLLCLAGLVFVSEAGPTGTGESKCPLMVKVLDAVRGSPAINVAVHVFRKAADDT
WEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDS
GPRRYTIAALLSPYSYSTTAVVTNPKE
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  Blast E-value cutoff:
BDBM50308499
n/a
NameBDBM50308499
Synonyms:CHEMBL602722 | Ethyl 5-(4-chlorobenzoyl)-4-phenylthiazol-2-ylcarbamate | cid_7315332
TypeSmall organic molecule
Emp. Form.C19H15ClN2O3S
Mol. Mass.386.852
SMILESCCOC(=O)Nc1nc(c(s1)C(=O)c1ccc(Cl)cc1)-c1ccccc1
Structure
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