| Reaction Details |
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 | Report a problem with these data |
| Target | Free fatty acid receptor 4 |
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| Ligand | BDBM286163 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | AlphaScreen SureFire Assay |
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| Temperature | 298.15±n/a K |
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| EC50 | 1880±n/a nM |
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| Comments | extracted |
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| Citation |  Shi, Y; Cheng, PT; Wang, Y; Wu, SC; Zhang, H Bicyclo [2.2.1] acid GPR120 modulators US Patent US9518000 Publication Date 12/13/2016 |
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| More Info.: | Get all data from this article, Assay Method |
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| Free fatty acid receptor 4 |
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| Name: | Free fatty acid receptor 4 |
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| Synonyms: | FFAR4 | FFAR4_HUMAN | G-protein coupled receptor 120 | G-protein coupled receptor 129 | G-protein coupled receptor GT01 | G-protein coupled receptor PGR4 | GPR120 | GPR129 | O3FAR1 | Omega-3 fatty acid receptor 1 | PGR4 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 42256.91 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_1508994 |
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| Residue: | 377 |
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| Sequence: | MSPECARAAGDAPLRSLEQANRTRFPFFSDVKGDHRLVLAAVETTVLVLIFAVSLLGNVC
ALVLVARRRRRGATACLVLNLFCADLLFISAIPLVLAVRWTEAWLLGPVACHLLFYVMTL
SGSVTILTLAAVSLERMVCIVHLQRGVRGPGRRARAVLLALIWGYSAVAALPLCVFFRVV
PQRLPGADQEISICTLIWPTIPGEISWDVSFVTLNFLVPGLVIVISYSKILQTSEHLLDA
RAVVTHSEITKASRKRLTVSLAYSESHQIRVSQQDFRLFRTLFLLMVSFFIMWSPIIITI
LLILIQNFKQDLVIWPSLFFWVVAFTFANSALNPILYNMTLCRNEWKKIFCCFWFPEKGA
ILTDTSVKRNDLSIISG
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| BDBM286163 |
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| n/a |
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| Name | BDBM286163 |
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| Synonyms: | 4-(4-(2-chloro-3,6- difluorobenzyl- oxy)bicyclo [2.2.1]heptan- 1-yl)butanoic acid | US9518000, Example 56 |
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| Type | Small organic molecule |
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| Emp. Form. | C18H21ClF2O3 |
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| Mol. Mass. | 358.807 |
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| SMILES | OC(=O)CCCC12CCC(CC1)(C2)OCc1c(F)ccc(F)c1Cl |
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| Structure | 
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