| Reaction Details |
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 | Report a problem with these data |
| Target | Acetyltransferase, GNAT family |
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| Ligand | BDBM152708 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Eis Ban Inhibition Assay |
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| pH | 8±n/a |
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| IC50 | >2.00e+5±n/a nM |
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| Comments | extracted |
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| Citation |  Green, KD; Biswas, T; Chang, C; Wu, R; Chen, W; Janes, BK; Chalupska, D; Gornicki, P; Hanna, PC; Tsodikov, OV; Joachimiak, A; Garneau-Tsodikova, S Biochemical and structural analysis of an Eis family aminoglycoside acetyltransferase from bacillus anthracis. Biochemistry54:3197-206 (2015) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Acetyltransferase, GNAT family |
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| Name: | Acetyltransferase, GNAT family |
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| Synonyms: | Eis_Ban acetyltransferase (Eis_Ban) |
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| Type: | Protein |
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| Mol. Mass.: | 45469.21 |
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| Organism: | Bacillus anthracis str. Sterne |
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| Description: | Q81P65 |
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| Residue: | 385 |
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| Sequence: | MNVIRLKEDKFREALRLSEYAFQYKVDEDRLQQQITKMKESHEVYGIMEGENLAAKLHLI
PFHIYIGKEKFKMGGVAGVATYPEYRRSGYVKELLQHSLQTMKKDGYTVSMLHPFAVSFY
RKYGWELCANLLVCHMTKSDLVMKKQVNGTVKRFNKESHPEEVEKLYETFAELFSGMLVR
NEKWWLQAVYDDLTLAIYYDENQTAAGYMLYKIENYKMTVEEFVPLHNEARNGLWNFICQ
HDSMIKDLEMTVSENEPLLYTLQEPRVKTEIKPYFMGRIVDVEQFLKQYELNWNNVQQEV
ILHITDSFAQWNNITVRIANHEITIIEEPIDKGIKLDINALSTILFGYRRPLELNELELI
SGSEEEIRAFESVVPVRKPFIYDFF
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| BDBM152708 |
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| n/a |
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| Name | BDBM152708 |
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| Synonyms: | 3-Chloro-N-[3-(diethylamino)propyl]-1-benzothiophene-2-carboxamide (3) |
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| Type | Small organic molecule |
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| Emp. Form. | C16H21ClN2OS |
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| Mol. Mass. | 324.869 |
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| SMILES | CCN(CC)CCCNC(=O)c1sc2ccccc2c1Cl |
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| Structure | 
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