| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Cannabinoid receptor 1 |
|---|
| Ligand | BDBM181246 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | CB1 Receptor Binding Protocol |
|---|
| Temperature | 303.15±n/a K |
|---|
| Ki | 2.33±0.09 nM |
|---|
| Comments | extracted |
|---|
| Citation |  Moore, II, BM; Bhattacharjee, H; Mustafa, S Tri-aryl/heteroaromatic cannabinoids and use thereof US Patent US9139546 Publication Date 9/22/2015 |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Cannabinoid receptor 1 |
|---|
| Name: | Cannabinoid receptor 1 |
|---|
| Synonyms: | CANN6 | CANNABINOID CB1 | CB-R | CB1 | CNR | CNR1 | CNR1_HUMAN | Cannabinoid CB1 receptor | Cannabinoid receptor | Cannabinoid receptor 1 (CB1) | Cannabinoid receptor 1 (brain) |
|---|
| Type: | G Protein-Coupled Receptor (GPCR) |
|---|
| Mol. Mass.: | 52868.96 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | P21554 |
|---|
| Residue: | 472 |
|---|
| Sequence: | MKSILDGLADTTFRTITTDLLYVGSNDIQYEDIKGDMASKLGYFPQKFPLTSFRGSPFQE
KMTAGDNPQLVPADQVNITEFYNKSLSSFKENEENIQCGENFMDIECFMVLNPSQQLAIA
VLSLTLGTFTVLENLLVLCVILHSRSLRCRPSYHFIGSLAVADLLGSVIFVYSFIDFHVF
HRKDSRNVFLFKLGGVTASFTASVGSLFLTAIDRYISIHRPLAYKRIVTRPKAVVAFCLM
WTIAIVIAVLPLLGWNCEKLQSVCSDIFPHIDETYLMFWIGVTSVLLLFIVYAYMYILWK
AHSHAVRMIQRGTQKSIIIHTSEDGKVQVTRPDQARMDIRLAKTLVLILVVLIICWGPLL
AIMVYDVFGKMNKLIKTVFAFCSMLCLLNSTVNPIIYALRSKDLRHAFRSMFPSCEGTAQ
PLDNSMGDSDCLHKHANNAASVHRAAESCIKSTVKIAKVTMSVSTDTSAEAL
|
|
|
|---|
| BDBM181246 |
|---|
| n/a |
|---|
| Name | BDBM181246 |
|---|
| Synonyms: | US9139546, 44 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C19H16Cl2O2S |
|---|
| Mol. Mass. | 379.3 |
|---|
| SMILES | CC(C)(c1cccs1)c1cc(O)c(c(O)c1)-c1cc(Cl)cc(Cl)c1 |
|---|
| Structure | 
|
|---|
Search and Browse
