| Reaction Details |
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 | Report a problem with these data |
| Target | Prostaglandin E2 receptor EP2 subtype |
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| Ligand | BDBM184625 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Radioligand Binding |
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| pH | 7.4±n/a |
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| Temperature | 277.15±n/a K |
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| IC50 | 1500±n/a nM |
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| EC50 | 944±n/a nM |
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| Comments | extracted |
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| Citation |  Donde, Y; Nguyen, JH; Kedzie, KM; Gil, DW; Donello, JE; Im, W Treatment of inflammatory bowel disease US Patent US9156810 Publication Date 10/13/2015 |
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| More Info.: | Get all data from this article, Assay Method |
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| Prostaglandin E2 receptor EP2 subtype |
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| Name: | Prostaglandin E2 receptor EP2 subtype |
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| Synonyms: | PE2R2_HUMAN | PGE receptor EP2 subtype | PTGER2 | Prostaglandin E2 | Prostaglandin E2 receptor | Prostaglandin E2 receptor EP4 subtype | Prostanoid EP2 Receptor |
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| Type: | Enzyme |
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| Mol. Mass.: | 39775.71 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P43116 |
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| Residue: | 358 |
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| Sequence: | MGNASNDSQSEDCETRQWLPPGESPAISSVMFSAGVLGNLIALALLARRWRGDVGCSAGR
RSSLSLFHVLVTELVFTDLLGTCLISPVVLASYARNQTLVALAPESRACTYFAFAMTFFS
LATMLMLFAMALERYLSIGHPYFYQRRVSRSGGLAVLPVIYAVSLLFCSLPLLDYGQYVQ
YCPGTWCFIRHGRTAYLQLYATLLLLLIVSVLACNFSVILNLIRMHRRSRRSRCGPSLGS
GRGGPGARRRGERVSMAEETDHLILLAIMTITFAVCSLPFTIFAYMNETSSRKEKWDLQA
LRFLSINSIIDPWVFAILRPPVLRLMRSVLCCRISLRTQDATQTSCSTQSDASKQADL
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| BDBM184625 |
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| n/a |
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| Name | BDBM184625 |
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| Synonyms: | US9156810, 44 |
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| Type | Small organic molecule |
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| Emp. Form. | C22H36O5 |
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| Mol. Mass. | 380.5182 |
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| SMILES | CCCCC[C@H](O)\C=C\[C@H]1[C@H](O)C(C)(C)C(=O)[C@@H]1C\C=C/CCCC(O)=O |
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| Structure | 
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