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TargetFatty acid-binding protein, liver
LigandBDBM50212873
Substrate/CompetitorBDBM60925
Meas. Tech.FABP1 Fluorescent Ligand Displacement Assay
Ki 52± 1 nM
Citation Huang, HMcIntosh, ALMartin, GGLandrock, DChung, SLandrock, KKDangott, LJLi, SKier, ABSchroeder, F FABP1: A Novel Hepatic Endocannabinoid and Cannabinoid Binding Protein. Biochemistry55:5243-55 (2016) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Fatty acid-binding protein, liver
Name:Fatty acid-binding protein, liver
Synonyms:FABPL_MOUSE | Fabp1 | Fabpl | Liver fatty acid binding protein (FABP1)
Type:Protein
Mol. Mass.:14247.91
Organism:Mus musculus (Mouse)
Description:n/a
Residue:127
Sequence:
MNFSGKYQLQSQENFEPFMKAIGLPEDLIQKGKDIKGVSEIVHEGKKIKLTITYGPKVVR
NEFTLGEECELETMTGEKVKAVVKLEGDNKMVTTFKGIKSVTELNGDTITNTMTLGDIVY
KRVSKRI
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BDBM50212873
BDBM60925
NameBDBM50212873
Synonyms:((2'-(5-ETHYL-3,4-DIPHENYL-1H-PYRAZOL-1-YL)-3-BIPHENYLYL)OXY)ACETIC ACID | BMS309403 | CHEMBL247920 | [2'-(5-Ethyl-3,4-diphenyl-pyrazol-1-yl)-biphenyl-3-yloxy]-acetic acid
TypeSmall organic molecule
Emp. Form.C31H26N2O3
Mol. Mass.474.5497
SMILESCCc1c(c(nn1-c1ccccc1-c1cccc(OCC(O)=O)c1)-c1ccccc1)-c1ccccc1
Structure
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