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TargetFatty acid-binding protein, liver
LigandBDBM21278
Substrate/Competitorn/a
Meas. Tech.FABP1 Fluorescent Ligand Displacement Assay
Ki 2.0e+3± 4e+2 nM
Citation Huang, HMcIntosh, ALMartin, GGLandrock, DChung, SLandrock, KKDangott, LJLi, SKier, ABSchroeder, F FABP1: A Novel Hepatic Endocannabinoid and Cannabinoid Binding Protein. Biochemistry55:5243-55 (2016) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Fatty acid-binding protein, liver
Name:Fatty acid-binding protein, liver
Synonyms:FABPL_MOUSE | Fabp1 | Fabpl | Liver fatty acid binding protein (FABP1)
Type:Protein
Mol. Mass.:14247.91
Organism:Mus musculus (Mouse)
Description:n/a
Residue:127
Sequence:
MNFSGKYQLQSQENFEPFMKAIGLPEDLIQKGKDIKGVSEIVHEGKKIKLTITYGPKVVR
NEFTLGEECELETMTGEKVKAVVKLEGDNKMVTTFKGIKSVTELNGDTITNTMTLGDIVY
KRVSKRI
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BDBM21278
n/a
NameBDBM21278
Synonyms:5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide | Acomplia | CHEMBL111 | CHEMBL558598 | RIMONABANT HYDROCHLORIDE | Rimonabant | SR 141716A | SR141716 | SR141716A | [3H]Rimonabant | [3H]SR141716A
TypeSmall organic molecule
Emp. Form.C22H21Cl3N4O
Mol. Mass.463.787
SMILESCc1c(nn(c1-c1ccc(Cl)cc1)-c1ccc(Cl)cc1Cl)C(=O)NN1CCCCC1
Structure
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