| Reaction Details |
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 | Report a problem with these data |
| Target | Opioid growth factor receptor-like protein 1 |
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| Ligand | BDBM199352 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Radioligand Dose-Displacement Binding Assay |
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| pH | 7.4±n/a |
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| Temperature | 323.15±n/a K |
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| Ki | 187.98±7.09 nM |
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| Comments | extracted |
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| Citation |  Kyle, DJ; Tafesse, L Buprenorphine analogs US Patent US9221831 Publication Date 12/29/2015 |
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| More Info.: | Get all data from this article, Assay Method |
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| Opioid growth factor receptor-like protein 1 |
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| Name: | Opioid growth factor receptor-like protein 1 |
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| Synonyms: | OGFRL1 | OGRL1_HUMAN | Opioid Receptor-Like Receptor (ORL-1) | Opioid growth factor receptor-like protein 1 (ORL-1) | Opioid growth factor receptor-like protein 1 (ORL1) | Opioid receptor-like (ORL-1) | Opioid receptor-like (ORL1) | Opioid receptor-like protein 1 (OGL1) | Opioid receptor-like receptor (ORL1) |
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| Type: | Protein |
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| Mol. Mass.: | 51247.53 |
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| Organism: | Homo sapiens (Human) |
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| Description: | Q5TC84 |
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| Residue: | 451 |
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| Sequence: | MGNLLGGVSFREPTTVEDCDSTWQTDSEPEPEEPGPGGGSEGPGQESEQPAQPPEQAGGR
PGASPAPDEDAEAAGAEQGGDSTEATAKPKRSFYAARDLYKYRHQYPNFKDIRYQNDLSN
LRFYKNKIPFKPDGVYIEEVLSKWKGDYEKLEHNHTYIQWLFPLREQGLNFYAKELTTYE
IEEFKKTKEAIRRFLLAYKMMLEFFGIKLTDKTGNVARAVNWQERFQHLNESQHNYLRIT
RILKSLGELGYESFKSPLVKFILHEALVENTIPNIKQSALEYFVYTIRDRRERRKLLRFA
QKHYTPSENFIWGPPRKEQSEGSKAQKMSSPLASSHNSQTSMHKKAKDSKNSSSAVHLNS
KTAEDKKVAPKEPVEETDRPSPEPSNEAAKPRNTEKDSNAENMNSQPEKTVTTPTEKKES
VSPENNEEGGNDNQDNENPGNTNCHDVVLVQ
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| BDBM199352 |
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| n/a |
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| Name | BDBM199352 |
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| Synonyms: | US9221831, 17 |
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| Type | Small organic molecule |
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| Emp. Form. | C30H36N2O4 |
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| Mol. Mass. | 488.6178 |
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| SMILES | CO[C@]12CC[C@@]3(C[C@@H]1COCc1ccccc1)[C@H]1Cc4ccc(NC(C)=O)c5O[C@@H]2[C@]3(CCN1C)c45 |r,TLB:8:7:30.29:4.3| |
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| Structure | 
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