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TargetCHK1_Kinase
LigandBDBM225375
Substrate/Competitorn/a
Meas. Tech.33P-Radiometric_Method1
Ki 0.299±n/a nM
Citation D3R DD Abbott CHK1 Kinase D3R  221 Publication Date 6/30/2015
More Info.:Get all data from this article,  Assay Method
 
CHK1_Kinase
Name:CHK1_Kinase
Synonyms:n/a
Type:n/a
Mol. Mass.:32109.16
Organism:Homo sapiens (Human)
Description:n/a
Residue:279
Sequence:
AVPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKRAVDCPENIKKEICINKM
LNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYL
HGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKR
REFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLAL
LHKILVENPSARITIPDIKKDRWYNKPLKKGAKRPRVTS
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  Blast E-value cutoff:
BDBM225375
n/a
NameBDBM225375
Synonyms:Chk1_144
TypeSmall Organic Molecule
Emp. Form.C23H19N3O3
Mol. Mass.385.4153
SMILESCOc1cc2Cc3c(n[nH]c3-c3ccc(nc3)-c3ccc(O)cc3)-c2cc1OC
Structure
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