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TargetUrokinase-type plasminogen activator [179-424,C299A,N323Q]
LigandBDBM92315
Substrate/Competitorn/a
Meas. Tech.Photometric_Method1
Ki 777±n/a nM
Citation D3R, DD Abbott Urokinase D3R D3R Publication Date 6/30/2015
More Info.:Get all data from this article,  Assay Method
 
Urokinase-type plasminogen activator [179-424,C299A,N323Q]
Name:Urokinase-type plasminogen activator [179-424,C299A,N323Q]
Synonyms:PLAU | UROK_HUMAN | Urokinase
Type:n/a
Mol. Mass.:27687.84
Organism:Homo sapiens (Human)
Description:P00749[179-424,C299A,N323Q]
Residue:246
Sequence:
IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVY
LGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTI
ALPSMYNDPQFGTSCEITGFGKEQSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTK
MLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPW
IRSHTK
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BDBM92315
n/a
NameBDBM92315
Synonyms:uPa_38
Typen/a
Emp. Form.C25H27BrN2O3
Mol. Mass.483.397
SMILESCCOc1cc(OCC)c(\C=C\c2cc(Br)c3cc(ccc3c2)C(N)=N)cc1OCC
Structure
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