| Reaction Details |
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 | Report a problem with these data |
| Target | Hexokinase-4 |
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| Ligand | BDBM239066 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Activation Assay |
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| pH | 7.1±n/a |
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| EC50 | 2000±n/a nM |
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| Citation |  Kang, X; Long, W; Ma, C; Wang, Y; Shen, X; Hu, Y; Tan, F; Wang, Y Compound for increasing kinase active and application thereof US Patent US9409900 Publication Date 8/9/2016 |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Hexokinase-4 |
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| Name: | Hexokinase-4 |
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| Synonyms: | Gck | Gk | Glucokinase | HK IV | HK4 | HXK4_MOUSE | Hexokinase-4 | Hexokinase-D |
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| Type: | Enzyme |
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| Mol. Mass.: | 52075.40 |
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| Organism: | Mus musculus (Mouse) |
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| Description: | P52792 |
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| Residue: | 465 |
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| Sequence: | MLDDRARMEATKKEKVEQILAEFQLQEEDLKKVMSRMQKEMDRGLKLETHQEASVKMLPT
YVRSTPEGSEVGDFLSLDLGGTNFRVMLVKVGEGEAGQWSVKTKHQMYSIPEDAMTGTAE
MLFDYISECISDFLDKHQMKHKKLPLGFTFSFPVRHEDIDKGILLNWTKGFKASGAEGNN
IVGLLRDAIKRRGDFEMDVVAMVNDTVATMISCYYEDRQCEVGMIVGTGCNACYMEEMQN
VELVEGDEGRMCVNTEWGAFGNSGELDEFLLEYDRMVDESSVNPGQQLYEKIIGGKYMGE
LVRLVLLKLVEENLLFHGEASEQLRTRGAFETRFVSQVESDSGDRRQILNILSTLGLRPS
VADCDIVRRACESVSTRAAHMCSAGLAGVINRMRESRSEDVMRITVGVDGSVYKLHPSFK
ERFHASVRRLTPNCEITFIESEEGSGRGAALVSAVACKKACMLGQ
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| BDBM239066 |
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| n/a |
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| Name | BDBM239066 |
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| Synonyms: | US9409900, 13 |
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| Type | Small organic molecule |
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| Emp. Form. | C21H22N4O4S2 |
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| Mol. Mass. | 458.554 |
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| SMILES | Cc1cnc(Nc2ccc(Oc3ccc(nc3)S(C)(=O)=O)c(CN3CCCC3=O)c2)s1 |
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| Structure | 
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