| Reaction Details |
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 | Report a problem with these data |
| Target | Cyclin-dependent kinase 5 activator 1 [99-307] |
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| Ligand | BDBM357015 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Caliper Kinase Assay |
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| IC50 | 50000±n/a nM |
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| Citation |  Johnson, JA; Lloyd, J; Finlay, H; Neels, J; Dhondi, NK; Gunaga, P; Banerjee, A; Adisechan, A Quinazolines as potassium ion channel inhibitors US Patent US10676460 Publication Date 6/9/2020 |
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| More Info.: | Get all data from this article, Assay Method |
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| Cyclin-dependent kinase 5 activator 1 [99-307] |
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| Name: | Cyclin-dependent kinase 5 activator 1 [99-307] |
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| Synonyms: | CD5R1_HUMAN | CDK5R | CDK5R1 | Cyclin-Dependent Kinase 5 Activator | Cyclin-dependent kinase 5 activator 1, p25 | NCK5A | TPKII regulatory subunit | p25 |
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| Type: | Enzyme Subunit |
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| Mol. Mass.: | 23250.56 |
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| Organism: | Homo sapiens (Human) |
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| Description: | Q15078 aa 99-307 |
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| Residue: | 209 |
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| Sequence: | AQPPPAQPPAPPASQLSGSQTGGSSSVKKAPHPAVTSAGTPKRVIVQASTSELLRCLGEF
LCRRCYRLKHLSPTDPVLWLRSVDRSLLLQGWQDQGFITPANVVFLYMLCRDVISSEVGS
DHELQAVLLTCLYLSYSYMGNEISYPLKPFLVESCKEAFWDRCLSVINLMSSKMLQINAD
PHYFTQVFSDLKNESGQEDKKRLLLGLDR
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| BDBM357015 |
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| n/a |
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| Name | BDBM357015 |
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| Synonyms: | US10214511, Example 19 | US10676460, Example 19 |
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| Type | Small organic molecule |
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| Emp. Form. | C20H15ClN4 |
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| Mol. Mass. | 346.813 |
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| SMILES | Clc1nc(NCc2ccccn2)c2c(cccc2n1)-c1ccccc1 |
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| Structure | 
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